Drug discovery targeting human 5-HT(2C) receptors: residues S3.36 and Y7.43 impact ligand-binding pocket structure via hydrogen bond formation (Q35573424)

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scientific article published on 12 October 2011

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English	Drug discovery targeting human 5-HT(2C) receptors: residues S3.36 and Y7.43 impact ligand-binding pocket structure via hydrogen bond formation	scientific article published on 12 October 2011

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

8 August 2017

Drug discovery targeting human 5-HT(2C) receptors: residues S3.36 and Y7.43 impact ligand-binding pocket structure via hydrogen bond formation (English)

1 reference

Europe PubMed Central

PubMed publication ID

8 August 2017

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based on heuristic

inferred from title

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based on heuristic

inferred from title

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based on heuristic

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Tania C Cordova-Sintjago

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Tania C Cordova-Sintjago

2

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author name string

Clinton E Canal

1

1 reference

Europe PubMed Central

PubMed publication ID

8 August 2017

Nancy Y Villa

3

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Europe PubMed Central

PubMed publication ID

8 August 2017

Li-Juan Fang

4

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Europe PubMed Central

PubMed publication ID

8 August 2017

Raymond G Booth

5

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Europe PubMed Central

PubMed publication ID

8 August 2017

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publication date

12 October 2011

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Europe PubMed Central

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8 August 2017

European Journal of Pharmacology

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Europe PubMed Central

PubMed publication ID

8 August 2017

673

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Europe PubMed Central

PubMed publication ID

8 August 2017

1-3

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Europe PubMed Central

PubMed publication ID

8 August 2017

1-12

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Europe PubMed Central

PubMed publication ID

8 August 2017

Structure and function of an irreversible agonist-β(2) adrenoceptor complex

1 reference

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Structure of a nanobody-stabilized active state of the β(2) adrenoceptor

1 reference

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1 reference

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Multiplicity of mechanisms of serotonin receptor signal transduction

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1 reference

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1 reference

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Agonist high and low affinity state ratios predict drug intrinsic activity and a revised ternary complex mechanism at serotonin 5-HT(2A) and 5-HT(2C) receptors

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Assessment of the roles of serines 5.43(239) and 5.46(242) for binding and potency of agonist ligands at the human serotonin 5-HT2A receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/22020288

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.EJPHAR.2011.10.006

1 reference

Europe PubMed Central

PubMed publication ID

8 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

8 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

8 August 2017

ResearchGate publication ID

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