CC12, a high-affinity ligand for [3H]cimetidine binding, is an improgan antagonist (Q35842760)

10 August 2017

CC12, a high-affinity ligand for [3H]cimetidine binding, is an improgan antagonist (English)

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10 August 2017

Lindsay B Hough

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10 August 2017

Julia W Nalwalk

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10 August 2017

James G Phillips

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10 August 2017

Brian Kern

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10 August 2017

Zhixing Shan

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10 August 2017

Mark P Wentland

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10 August 2017

Iwan J P de Esch

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10 August 2017

Elwin Janssen

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10 August 2017

Travis Barr

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10 August 2017

Rebecca Stadel

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10 August 2017

20 January 2007

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52

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5

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1244-1255

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describes a project that uses

10 August 2017

ImageQuant

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11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC1892205/fullTextXML

inferred from PubMed Central ID database lookup

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Antinociceptive activity of chemical congeners of improgan: optimization of side chain length leads to the discovery of a new, potent, non-opioid analgesic

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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Improgan, a cimetidine analog, induces morphine-like antinociception in opioid receptor-knockout mice

11 August 2018

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Circuitry underlying antiopioid actions of orphanin FQ in the rostral ventromedial medulla

11 August 2018

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11 August 2018

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The selective cannabinoid antagonist SR 141716A blocks cannabinoid-induced antinociception in rats

11 August 2018

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11 August 2018

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11 August 2018

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11 August 2018

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Characterization of the antinociceptive properties of cimetidine and a structural analog.

11 August 2018

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In vivo characterization of a specific cannabinoid receptor antagonist (SR141716A): inhibition of delta 9-tetrahydrocannabinol-induced responses and apparent agonist activity

11 August 2018

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Modulation of cannabinoid-induced antinociception after intracerebroventricular versus intrathecal administration to mice: possible mechanisms for interaction with morphine.

11 August 2018

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3H-cimetidine and the H2-receptor

11 August 2018

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Imidazole derivatives. Histidine decarboxylase inhibitors

11 August 2018

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Imidazole derivatives—A new class of microsomal enzyme inhibitors

11 August 2018

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Effects of some GABA-mimetic drugs on the antinociceptive activity of morphine and beta-endorphin in rats

11 August 2018

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12 December 2020

Cannabinoid-improgan cross-tolerance: Improgan is a cannabinomimetic analgesic lacking affinity at the cannabinoid CB1 receptor

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12 December 2020

Cannabinoid agonist signal transduction in rat brain: comparison of cannabinoid agonists in receptor binding, G-protein activation, and adenylyl cyclase inhibition.

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12 December 2020

Antinociceptive activity of derivatives of improgran and burimamide

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12 December 2020

Antagonism of an indirectly acting agonist: Block by propranolol and sotalol of the action of tyramien on rat heart

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12 December 2020

Characterization of histamine receptors in isolated pig basilar artery by functional and radioligand binding studies

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12 December 2020

Histamine receptors in an experimental mammary carcinoma

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12 December 2020

Binding of [3H]cimetidine to rat brain tissue

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12 December 2020

10.1016/J.NEUROPHARM.2007.01.004

Identifiers

DOI

1 reference

10 August 2017

1 reference

10 August 2017

PubMed publication ID

17336343

1 reference