Binding and functional properties of hexocyclium and sila-hexocyclium derivatives to muscarinic receptor subtypes (Q35874770)

10 August 2017

Binding and functional properties of hexocyclium and sila-hexocyclium derivatives to muscarinic receptor subtypes (English)

1 reference

10 August 2017

Waelbroeck M

1

1 reference

10 August 2017

Camus J

2

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10 August 2017

Tastenoy M

3

1 reference

10 August 2017

Feifel R

4

1 reference

10 August 2017

Mutschler E

5

1 reference

10 August 2017

Tacke R

6

1 reference

10 August 2017

Strohmann C

7

1 reference

10 August 2017

Rafeiner K

8

1 reference

10 August 2017

Rodrigues de Miranda JF

9

1 reference

10 August 2017

Lambrecht G

10

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10 August 2017

language of work or name

English

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publication date

1 June 1994

1 reference

British Journal of Pharmacology

10 August 2017

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10 August 2017

112

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10 August 2017

2

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10 August 2017

505-514

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Protein measurement with the Folin phenol reagent

10 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Some quantitative uses of drug antagonists

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Characterization of muscarinic receptors mediating vasodilation in rat perfused kidney

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Pharmacological characterization of acetylcholine-stimulated [35S]-GTP gamma S binding mediated by human muscarinic m1-m4 receptors: antagonist studies

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

New functionally selective muscarinic agonists

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Muscarinic receptors--characterization, coupling and function

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Structure-activity relationships of unsaturated esters of arecaidine and dihydroarecaidine

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

The relative potencies of some agonists at M2 muscarinic receptors in guinea-pig ileum, atria and bronchi

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

o-Methoxy-sila-hexocyclium: a new quaternary M1-selective muscarinic antagonist

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

80% of muscarinic receptors expressed by the NB-OK 1 human neuroblastoma cell line show high affinity for pirenzepine and are comparable to rat hippocampus M1 receptors

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Method for comparing selectivities of unlabeled subpopulation-selective ligands: application to muscarinic receptors.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Binding and functional properties of antimuscarinics of the hexocyclium/sila-hexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Antagonist binding properties of five cloned muscarinic receptors expressed in CHO-K1 cells

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Affinity profiles of hexahydro-sila-difenidol analogues at muscarinic receptor subtypes

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Human HT-29 colon carcinoma cells contain muscarinic M3 receptors coupled to phosphoinositide metabolism.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Binding of selective antagonists to four muscarinic receptors (M1 to M4) in rat forebrain

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Hexocyclium derivatives with a high selectivity for smooth muscle muscarinic receptors

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Novel pharmacological profile of muscarinic receptors mediating contraction of the guinea-pig uterus

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Characterization of muscarinic M4 binding sites in rabbit lung, chicken heart, and NG108-15 cells

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Muscarinic receptor subtypes

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Antagonist binding profiles of five cloned human muscarinic receptor subtypes

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Different effects of muscarinic agonssts in rat superior cervical ganglion and hippocampal slices

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Selective inhibition of responses to carbachol and McN-A-343 in the rabbit vas deferens.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

4-DAMP analogues reveal heterogeneity of M1 muscarinic receptors

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

pA2 and receptor differentiation: a statistical analysis of competitive antagonism

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Stereochemical analogs of a muscarinic, ganglionic stimulant. 2. The cis and trans olefinic, epoxide, and cyclopropane analogs related to 4-[N-(3-chlorophenyl)carbamoyloxy]-2-butynyltrimethylammonium chloride

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

Pirenzepine distinguishes between different subclasses of muscarinic receptors

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

The effects of pH on the affinity of pirenzepine for muscarinic receptors in the guinea-pig ileum and rat fundus strip

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

The origin of acetylcholine released from guinea-pig intestine and longitudinal muscle strips.

24 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1910350

The Uptake of Atropine and Related Drugs by Intestinal Smooth Muscle of the Guinea-Pig in Relation to Acetylcholine Receptors

24 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1994.TB13102.X

Human gastric mucosa expresses glandular M3 subtype of muscarinic receptors

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1994.TB13102.X

Presynaptic muscarinic receptors mediating inhibition of neurogenic contractions in rabbit vas deferens are of the ganglionic M1-type

21 January 2018

1 reference

12 December 2020

Muscarinic receptors mediating acid secretion in isolated rat gastric parietal cells are of M3 type

1 reference

12 December 2020

Selective antagonists provide evidence that M1 muscarinic receptors may mediate carbachol-induced drinking in the rat

1 reference

12 December 2020

Selective labelling of muscarinic M1 receptors in calf superior cervical ganglia by [3H](+/-)-telenzepine

1 reference

12 December 2020

Characterization of muscarinic receptors in guinea-pig uterus

1 reference

12 December 2020

Characterization of the prejunctional muscarinic receptors mediating inhibition of evoked release of endogenous noradrenaline in rabbit isolated vas deferens

1 reference

12 December 2020

Cumulative dose-response curves. II. Technique for the making of dose-response curves in isolated organs and the evaluation of drug parameters

1 reference

12 December 2020

Sila-substitution--a useful strategy for drug design?

1 reference

12 December 2020

Muscarinic receptor heterogeneity in rat central nervous system. I. Binding of four selective antagonists to three muscarinic receptor subclasses: a comparison with M2 cardiac muscarinic receptors of the C type

1 reference

12 December 2020

Different antagonist binding properties of rat pancreatic and cardiac muscarinic receptors

1 reference

12 December 2020

Muscarinic M1- and M2-receptors mediating opposite effects on neuromuscular transmission in rabbit vas deferens

1 reference

12 December 2020

10.1111/J.1476-5381.1994.TB13102.X

Identifiers

DOI

1 reference

release_xd4pm4zy7zejlc3lr2lrzhjpie

10 August 2017

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/xd4pm4zy7zejlc3lr2lrzhjpie

24 November 2022

mapped directly with Wikidata item

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10 August 2017

PubMed publication ID

8075869

1 reference