Heterogeneity of thromboxane A2 (TP-) receptors: evidence from antagonist but not agonist potency measurements (Q35888653)

10 August 2017

Heterogeneity of thromboxane A2 (TP-) receptors: evidence from antagonist but not agonist potency measurements (English)

1 reference

10 August 2017

1 reference

P. M. Tymkewycz

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1364826

18 September 2022

R. L. Jones

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1364826

18 September 2022

N. H. Wilson

series ordinal

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1364826

18 September 2022

C. G. Marr

series ordinal

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1364826

18 September 2022

language of work or name

English

0 references

publication date

1 March 1991

1 reference

PMCID

1917959

full work available at URL

10 August 2017

https://europepmc.org/articles/PMC1917959

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1364826

https://europepmc.org/articles/PMC1917959?pdf=render

18 September 2022

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1364826

British Journal of Pharmacology

18 September 2022

published in

1 reference

10 August 2017

102

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10 August 2017

3

1 reference

10 August 2017

607-614

1 reference

Some quantitative uses of drug antagonists

10 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

UK-37, 248, a novel, selective thromboxane synthetase inhibitor with platelet anti-aggregatory and anti-thrombotic activity

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Antagonism of the thromboxane-sensitive contractile systems of the rabbit aorta, dog saphenous vein and guinea-pig trachea

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Binding of a radioiodinated 13-azapinane thromboxane antagonist to platelets: correlation with antiaggregatory activity in different species

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Vitamin K 2,3-epoxide reductase: the basis for stereoselectivity of 4-hydroxycoumarin anticoagulant activity

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

AH23848: a thromboxane receptor-blocking drug that can clarify the pathophysiologic role of thromboxane A2.

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Evidence for homogeneity of thromboxane A2 receptor using structurally different antagonists

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Peripheral 5-HT2-like receptors. Can they be classified with the available antagonists?

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

EP 171: a high affinity thromboxane A2-mimetic, the actions of which are slowly reversed by receptor blockade

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Competitive antagonism at thromboxane receptors in human platelets

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Characteristics of [3H]-GR 32191 binding to the thromboxane (TP) receptor of human platelets

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

GR32191, a highly potent and specific thromboxane A2 receptor blocking drug on platelets and vascular and airways smooth muscle in vitro

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

How should values of pA2 and affinity constants for pharmacological competitive antagonists be estimated?

11 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1917959

Aggregation of Blood Platelets by Adenosine Diphosphate and its Reversal

11 July 2018

1 reference

Crossref

https://api.crossref.org/works/10.1111%2FJ.1476-5381.1991.TB12220.X

Prostaglandin E2: effects on aggregation, shape change and cyclic AMP of rat platelets

21 January 2018

1 reference

12 December 2020

Interactions of thromboxane A2 analogs and prostaglandins in isolated dog arteries

1 reference

12 December 2020

Effect of Prostaglandin E2 and Aspirin on the Secondary Aggregation of Human Platelets

1 reference

12 December 2020

Investigation on a selective non-prostanoic thromboxane antagonist, BM 13.177, in human platelets

1 reference

12 December 2020

Synthesis of prostanoids with bicyclo[2.2.1]heptane, bicyclo[3.1.1]heptane, and bicyclo[2.2.2]octane ring systems. Activities of 15-hydroxy epimers on human platelets

1 reference

12 December 2020

Pharmacologic characterization of human and canine thromboxane A2/prostaglandin H2 receptors in platelets and blood vessels: evidence for different receptors

1 reference

12 December 2020

Effects of the thromboxane receptor antagonist SK&F 88046 in the canine, monkey and human coronary vasculature

1 reference

12 December 2020

10.1111/J.1476-5381.1991.TB12220.X

Identifiers

DOI

1 reference

10 August 2017

1 reference

10 August 2017

1 reference

PMCID

1917959