Centrally active 5-HT receptor agonists and antagonists (Q35942133)

11 August 2017

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title

Centrally active 5-HT receptor agonists and antagonists (English)

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11 August 2017

D. N. Middlemiss

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1553108

8 October 2022

M. D. Tricklebank

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1553108

8 October 2022

language of work or name

English

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=1553108

8 October 2022

publication date

1 January 1992

1 reference

Neuroscience & Biobehavioral Reviews

11 August 2017

published in

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11 August 2017

volume

16

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11 August 2017

issue

1

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11 August 2017

page(s)

75-82

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[3H]zacopride: ligand for the identification of 5-HT3 recognition sites

11 August 2017

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The 5-HT1 receptor agonist RU-24969 decreases 5-hydroxytryptamine (5-HT) release and metabolism in the rat frontal cortex in vitro and in vivo

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Selective 5HT-2 antagonists inhibit serotonin stimulated phosphatidylinositol metabolism in cerebral cortex

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Neuroanatomical sites of action of 5-HT3 receptor agonist and antagonists for alteration of aversive behaviour in the mouse

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Possible benefit of GR43175, a novel 5-HT1-like receptor agonist, for the acute treatment of severe migraine

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A 5-HT receptor in the central nervous system, positively coupled with adenylate cyclase, is antagonized by ICS 205 930.

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Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites

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(+/-)[125Iodo] cyanopindolol, a new ligand for beta-adrenoceptors: identification and quantitation of subclasses of beta-adrenoceptors in guinea pig.

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NAN-190: an arylpiperazine analog that antagonizes the stimulus effects of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT).

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7 January 2021

Arylpiperazine derivatives as high-affinity 5-HT1A serotonin ligands

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7 January 2021

Molecular biology of 5-HT receptors

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7 January 2021

Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes

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7 January 2021

Mixed agonist/antagonist properties of NAN-190 at 5-HT1A receptors: behavioural and in vivo brain microdialysis studies.

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7 January 2021

Functional correlates of serotonin 5-HT1 recognition sites

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Characterization of the 5-HT1B recognition site in rat brain: binding studies with (-)[125I]iodocyanopindolol

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Species differences in the pharmacology of terminal 5-HT autoreceptors in mammalian brain

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Serotonin receptors in the human brain. I. Characterization and autoradiographic localization of 5-HT1A recognition sites. Apparent absence of 5-HT1B recognition sites

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5-HT1D receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in calf substantia nigra

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7 January 2021

The potential anxiolytic activity of GR38032F, a 5-HT3-receptor antagonist

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7 January 2021

Evidence that mCPP may have behavioural effects mediated by central 5-HT1C receptors

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7 January 2021

Evidence that hypophagia induced by mCPP and TFMPP requires 5-HT1C and 5-HT1B receptors; hypophagia induced by RU 24969 only requires 5-HT1B receptors

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7 January 2021

5-HT1B agonists induce anorexia at a postsynaptic site

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7 January 2021

Anxiogenic-like effects of mCPP and TFMPP in animal models are opposed by 5-HT1C receptor antagonists

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7 January 2021

1-(m-chlorophenyl)-biguanide, a potent high affinity 5-HT3 receptor agonist.

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7 January 2021

Identification and distribution of 5-HT3 receptors in rat brain using radioligand binding

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MK-212 increases rat plasma ACTH concentration by activation of the 5-HT1C receptor subtype.

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7 January 2021

Serotonin 5-HT2 receptors: two states versus two subtypes

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Receptor binding profile of R 41 468, A novel antagonist at 5-HT2 receptors

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7 January 2021

Differentiation of 5-hydroxytryptamine2 receptor subtypes using 125I-R-(-)2,5-dimethoxy-4-iodo-phenylisopropylamine and 3H-ketanserin.

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7 January 2021

Molecular size of the 5-HT3 receptor solubilized from NCB 20 cells

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7 January 2021

8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

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7 January 2021

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MDL 72832: a potent and stereoselective ligand at central and peripheral 5-HT1A receptors

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7 January 2021

Characterization of MDL 73005EF as a 5-HT1A selective ligand and its effects in animal models of anxiety: comparison with buspirone, 8-OH-DPAT and diazepam

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7 January 2021

Biochemical and pharmacological characterization of CGS 12066B, a selective serotonin-1B agonist

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7 January 2021

The binding of serotonergic ligands to the porcine choroid plexus: characterization of a new type of serotonin recognition site

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7 January 2021

Quantitative autoradiographic mapping of serotonin receptors in the rat brain. I. Serotonin-1 receptors

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7 January 2021

Discrimination of multiple [3H]5-hydroxytryptamine binding sites by the neuroleptic spiperone in rat brain

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7 January 2021

Sumatriptan (GR 43175) interacts selectively with 5-HT1B and 5-HT1D binding sites

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7 January 2021

Interaction of arylpiperazines with 5-HT1A, 5-HT1B, 5-HT1C and 5-HT1D receptors: do discriminatory 5-HT1B receptor ligands exist?

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7 January 2021

5-HT1 and 5-HT2 binding properties of derivatives of the hallucinogen 1-(2,5-dimethoxyphenyl)-2-aminopropane (2,5-DMA).

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7 January 2021

The discriminative stimulus properties of 2,5-dimethoxy-4-methylamphetamine (DOM): differentiation from amphetamine

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7 January 2021

Effect of acute and chronic MDL 73,147EF, a 5-HT3 receptor antagonist, on A9 and A10 dopamine neurons

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7 January 2021

Radioligand binding evidence implicates the brain 5-HT2 receptor as a site of action for LSD and phenylisopropylamine hallucinogens

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7 January 2021

Subtypes of 5-HT receptors

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7 January 2021

The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-propylamino)tetralin in the rat.

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7 January 2021

Pharmacological analysis of the behavioural and thermoregulatory effects of the putative 5-HT1 receptor agonist, RU 24969, in the rat

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7 January 2021

The concept of selectivity in 5-HT receptor research

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7 January 2021

The (S)-isomer of [3H]zacopride labels 5-HT3 receptors with high affinity in rat brain.

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7 January 2021

Interactions of isamoltane (CGP 361A), an anxiolytic phenoxypropanolamine derivative, with 5-HT1 receptor subtypes in the rat brain

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7 January 2021

BMY 7378, a buspirone analog with high affinity, selectivity and low intrinsic activity at the 5-HT1A receptor in rat and guinea pig hippocampal membranes

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7 January 2021

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Identifiers

DOI

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11 August 2017

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