Hydrophobic Interactions Improve Selectivity to ERα for Ben-zothiophene SERMs (Q35949610)

11 August 2017

Hydrophobic Interactions Improve Selectivity to ERα for Ben-zothiophene SERMs (English)

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11 August 2017

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Michael J Chalmers

1

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11 August 2017

Yong Wang

2

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11 August 2017

Scott Novick

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11 August 2017

Masahiko Sato

4

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11 August 2017

Henry U Bryant

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11 August 2017

Chahrzad Montrose-Rafizdeh

6

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11 August 2017

Patrick R Griffin

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11 August 2017

Jeffrey A Dodge

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11 August 2017

1 March 2012

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ACS Medicinal Chemistry Letters

11 August 2017

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11 August 2017

3

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11 August 2017

3

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11 August 2017

207-210

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Ligand-dependent perturbation of the conformational ensemble for the GPCR β2 adrenergic receptor revealed by HDX.

11 August 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Differential hydrogen/deuterium exchange mass spectrometry analysis of protein-ligand interactions

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Unique ligand binding patterns between estrogen receptor alpha and beta revealed by hydrogen-deuterium exchange.

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Prediction of the tissue-specificity of selective estrogen receptor modulators by using a single biochemical method

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Benzopyrans are selective estrogen receptor beta agonists with novel activity in models of benign prostatic hyperplasia

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Molecular basis of agonism and antagonism in the oestrogen receptor

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Cloning of a novel receptor expressed in rat prostate and ovary

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3349201

Structure-activity relationships of selective estrogen receptor modulators: modifications to the 2-arylbenzothiophene core of raloxifene

2 October 2017

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PubMed

https://pubmed.ncbi.nlm.nih.gov/22582136

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML2002532

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11 August 2017

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11 August 2017

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