Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model. (Q36071373)

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20 February 2020

title

Aiming for allosterism: Evaluation of allosteric modulators of CB1 in a neuronal model (English)

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20 February 2020

5

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20 February 2020

author name string

Alex Straiker

1

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20 February 2020

José Mitjavila

2

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20 February 2020

Danielle Yin

3

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20 February 2020

Anne Gibson

4

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20 February 2020

publication date

23 July 2015

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20 February 2020

published in

Pharmacological Research

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20 February 2020

volume

99

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20 February 2020

page(s)

370-376

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Localization and production of peptide endocannabinoids in the rodent CNS and adrenal medulla

20 February 2020

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2 October 2017

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Identification and quantification of a new family of peptide endocannabinoids (Pepcans) showing negative allosteric modulation at CB1 receptors

2 October 2017

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Allosteric modulator ORG27569 induces CB1 cannabinoid receptor high affinity agonist binding state, receptor internalization, and Gi protein-independent ERK1/2 kinase activation

2 October 2017

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Monoacylglycerol lipase limits the duration of endocannabinoid-mediated depolarization-induced suppression of excitation in autaptic hippocampal neurons

2 October 2017

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2 October 2017

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2 October 2017

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PSNCBAM-1, a novel allosteric antagonist at cannabinoid CB1 receptors with hypophagic effects in rats

2 October 2017

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Allosteric modulation of the cannabinoid CB1 receptor

2 October 2017

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2 October 2017

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Modulation of Ca2+ channels by G-protein beta gamma subunits

2 October 2017

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2 October 2017

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2 October 2017

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2 October 2017

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11 July 2018

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Characterization and Partial Purification of AIM: A Plasma Protein That Induces Rat Cerebral Type 2 Astroglia from Bipotential Glial Progenitors

11 July 2018

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11 July 2018

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An allosteric model for benzodiazepine receptor function

23 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/26211948

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.PHRS.2015.07.017

1 reference

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20 February 2020

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20 February 2020

PubMed publication ID

26211948

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:26211948%20AND%20SRC:MED&resulttype=core&format=json