Diisothiocyanate derivatives as potent, insurmountable antagonists of P2Y6 nucleotide receptors. (Q36146795)

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27 December 2019

title

Diisothiocyanate derivatives as potent, insurmountable antagonists of P2Y6 nucleotide receptors (English)

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27 December 2019

5

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3

Zhan-Guo Gao

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27 December 2019

4

Ivar von Kügelgen

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1

Liaman K Mamedova

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27 December 2019

2

Bhalchandra V Joshi

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27 December 2019

language of work or name

English

0 references

publication date

1 May 2004

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27 December 2019

published in

Biochemical Pharmacology

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27 December 2019

volume

67

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27 December 2019

issue

9

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27 December 2019

page(s)

1763-1770

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Structural determinants of efficacy at A3 adenosine receptors: modification of the ribose moiety.

27 December 2019

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

P2Y6 nucleotide receptor activates PKC to protect 1321N1 astrocytoma cells against tumor necrosis factor-induced apoptosis

2 October 2017

1 reference

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N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors

2 October 2017

1 reference

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Tumor necrosis factor alpha-induced apoptosis in astrocytes is prevented by the activation of P2Y6, but not P2Y4 nucleotide receptors

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

Models and methods for studying insurmountable antagonism

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

Quantitation of the P2Y(1) receptor with a high affinity radiolabeled antagonist

2 October 2017

1 reference

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Purine and pyrimidine (P2) receptors as drug targets

2 October 2017

1 reference

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p53-Independent induction of Fas and apoptosis in leukemic cells by an adenosine derivative, Cl-IB-MECA.

2 October 2017

1 reference

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Differential coupling of the human P2Y(11) receptor to phospholipase C and adenylyl cyclase

2 October 2017

1 reference

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Expression of the P2Y6 purinergic receptor in human T cells infiltrating inflammatory bowel disease.

2 October 2017

1 reference

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Receptors for purines and pyrimidines

2 October 2017

1 reference

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Characterisation of subtypes of the P2X and P2Y families of ATP receptors in the foetal human heart

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

Cloning of a human purinergic P2Y receptor coupled to phospholipase C and adenylyl cyclase

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

Families of ion channels with two hydrophobic segments

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

Uridine nucleotide selectivity of three phospholipase C-activating P2 receptors: identification of a UDP-selective, a UTP-selective, and an ATP- and UTP-specific receptor

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

G protein-coupled receptors for ATP and other nucleotides: a new receptor family

2 October 2017

1 reference

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High affinity acylating antagonists for the A1 adenosine receptor: identification of binding subunit

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

Novel irreversible ligands specific for "peripheral" type benzodiazepine receptors: (+/-)-, (+)-, and (-)-1-(2-chlorophenyl)-N-(1-methylpropyl)-N- (2-isothiocyanatoethyl)-3-isoquinolinecarboxamide and 1-(2-isothiocyanatoethyl)-7-chloro-1,3-dihydro-5

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

2 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3413726

P2 purinoceptor-mediated control of rat cerebral (pial) microvasculature; contribution of P2X and P2Y receptors

2 October 2017

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15081875

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Expression of the human P2Y6 nucleotide receptor in normal placenta and gestational trophoblastic disease

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15081875

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Increase in cardiac P2X1-and P2Y2-receptor mRNA levels in congestive heart failure

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15081875

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BCP.2004.01.011

1 reference

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27 December 2019

1 reference

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27 December 2019

1 reference