Illuminating the activation mechanisms and allosteric properties of metabotropic glutamate receptors (Q36762520)

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25 February 2020

title

Illuminating the activation mechanisms and allosteric properties of metabotropic glutamate receptors (English)

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25 February 2020

4

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25 February 2020

Jean-Philippe Pin

6

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25 February 2020

Philippe Rondard

7

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25 February 2020

author name string

Etienne Doumazane

1

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25 February 2020

Pauline Scholler

2

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25 February 2020

Ludovic Fabre

3

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25 February 2020

Eric Trinquet

5

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25 February 2020

language of work or name

English

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publication date

4 March 2013

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Proceedings of the National Academy of Sciences of the United States of America

25 February 2020

published in

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25 February 2020

volume

110

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issue

15

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25 February 2020

page(s)

E1416-25

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Sequential inter- and intrasubunit rearrangements during activation of dimeric metabotropic glutamate receptor 1.

25 February 2020

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29 September 2017

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29 September 2017

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Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to GPCR oligomerization

29 September 2017

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Functioning of the dimeric GABA(B) receptor extracellular domain revealed by glycan wedge scanning.

29 September 2017

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Optical techniques to analyze real-time activation and signaling of G-protein-coupled receptors.

29 September 2017

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Activation of a dimeric metabotropic glutamate receptor by intersubunit rearrangement.

29 September 2017

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29 September 2017

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Night blindness-associated mutations in the ligand-binding, cysteine-rich, and intracellular domains of the metabotropic glutamate receptor 6 abolish protein trafficking

29 September 2017

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Structures of the extracellular regions of the group II/III metabotropic glutamate receptors

29 September 2017

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29 September 2017

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A novel constitutively active mutation in the second cytoplasmic loop of metabotropic glutamate receptor.

29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor

29 September 2017

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Characterization of [(3)H]-LY354740 binding to rat mGlu2 and mGlu3 receptors expressed in CHO cells using semliki forest virus vectors

29 September 2017

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Amino acids in the second and third intracellular loops of the parathyroid Ca2+-sensing receptor mediate efficient coupling to phospholipase C.

29 September 2017

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Pharmacological agents acting at subtypes of metabotropic glutamate receptors

29 September 2017

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Role of the second and third intracellular loops of metabotropic glutamate receptors in mediating dual signal transduction activation

29 September 2017

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Pharmacology and functions of metabotropic glutamate receptors

29 September 2017

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A modern ionotropic glutamate receptor with a K(+) selectivity signature sequence.

29 September 2017

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Activation switch in the transmembrane domain of metabotropic glutamate receptor.

5 September 2018

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A general method for the covalent labeling of fusion proteins with small molecules in vivo

5 September 2018

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Coupling of agonist binding to effector domain activation in metabotropic glutamate-like receptors

5 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23487753

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

The non-competitive antagonists 2-methyl-6-(phenylethynyl)pyridine and 7-hydroxyiminocyclopropan[b]chromen-1a-carboxylic acid ethyl ester interact with overlapping binding pockets in the transmembrane region of group I metabotropic glutamate recepto

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23487753

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.1215615110

1 reference

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25 February 2020

0 references

1 reference

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25 February 2020

PubMed publication ID

23487753

1 reference