Investigating the kinetic mechanism of inhibition of elongation factor 2 kinase by NH125: evidence of a common in vitro artifact (Q36903990)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22352903%20AND%20SRC:MED&resulttype=core&format=json

23 January 2020

title

Investigating the kinetic mechanism of inhibition of elongation factor 2 kinase by NH125: evidence of a common in vitro artifact (English)

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23 January 2020

4

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23 January 2020

Kıvanç Görgülü

7

1 reference

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23 January 2020

Kıvanç Görgülü

8

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23 January 2020

author name string

Ashwini K Devkota

1

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23 January 2020

Clint D J Tavares

2

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23 January 2020

Mangalika Warthaka

3

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23 January 2020

Kyle D Marshall

5

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23 January 2020

Tamer S Kaoud

6

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23 January 2020

Bulent Ozpolat

9

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23 January 2020

Kevin N Dalby

10

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23 January 2020

language of work or name

English

0 references

publication date

5 March 2012

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23 January 2020

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23 January 2020

volume

51

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23 January 2020

issue

10

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23 January 2020

page(s)

2100-2112

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1-Benzyl-3-cetyl-2-methylimidazolium iodide (NH125) induces phosphorylation of eukaryotic elongation factor-2 (eEF2): a cautionary note on the anticancer mechanism of an eEF2 kinase inhibitor

23 January 2020

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29 September 2017

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29 September 2017

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27 June 2018

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27 June 2018

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27 June 2018

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27 June 2018

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27 June 2018

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4 September 2018

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4 September 2018

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4 September 2018

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4 September 2018

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4 September 2018

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4 September 2018

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4 September 2018

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12 December 2020

Autophagy and cancer therapy

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12 December 2020

Kinetic characterization of human JNK2alpha2 reaction mechanism using substrate competitive inhibitors

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12 December 2020

Identification and characterization of a potent antibacterial agent, NH125 against drug-resistant bacteria

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12 December 2020

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12 December 2020

Mechanism of elongation factor 2 (EF-2) inactivation upon phosphorylation. Phosphorylated EF-2 is unable to catalyze translocation

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12 December 2020

Increased activity of the eEF-2 specific, Ca2+ and calmodulin dependent protein kinase III during the S-phase in Ehrlich ascites cells

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Identifiers

DOI

10.1021/BI201787P

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22352903%20AND%20SRC:MED&resulttype=core&format=json

23 January 2020

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23 January 2020

1 reference

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