Sustained treatment with a 5-HT(2A) receptor agonist causes functional desensitization and reductions in agonist-labeled 5-HT(2A) receptors despite increases in receptor protein levels in rats (Q36962803)

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scientific article published on 07 June 2008

Language	Label	Description	Also known as
English	Sustained treatment with a 5-HT(2A) receptor agonist causes functional desensitization and reductions in agonist-labeled 5-HT(2A) receptors despite increases in receptor protein levels in rats	scientific article published on 07 June 2008

Statements

scholarly article

1 reference

Europe PubMed Central

17 August 2017

Sustained treatment with a 5-HT(2A) receptor agonist causes functional desensitization and reductions in agonist-labeled 5-HT(2A) receptors despite increases in receptor protein levels in rats (English)

1 reference

Europe PubMed Central

17 August 2017

desensitization

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based on heuristic

inferred from title

0 references

author name string

Ju Shi

1

1 reference

Europe PubMed Central

17 August 2017

Michelle Landry

2

1 reference

Europe PubMed Central

17 August 2017

Gonzalo A Carrasco

3

1 reference

Europe PubMed Central

17 August 2017

George Battaglia

4

1 reference

Europe PubMed Central

17 August 2017

Nancy A Muma

5

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Europe PubMed Central

17 August 2017

publication date

7 June 2008

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Europe PubMed Central

17 August 2017

Neuropharmacology

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Europe PubMed Central

17 August 2017

55

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Europe PubMed Central

17 August 2017

5

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Europe PubMed Central

17 August 2017

687-692

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Europe PubMed Central

17 August 2017

Agonist induced-phosphorylation of Galpha11 protein reduces coupling to 5-HT2A receptors.

1 reference

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Olanzapine increases RGS7 protein expression via stimulation of the Janus tyrosine kinase-signal transducer and activator of transcription signaling cascade.

1 reference

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Phosphorylation of Galpha11 protein contributes to agonist-induced desensitization of 5-HT2A receptor signaling

1 reference

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Evidence that 5-HT2A receptors in the hypothalamic paraventricular nucleus mediate neuroendocrine responses to (-)DOI

1 reference

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Paradoxical trafficking and regulation of 5-HT(2A) receptors by agonists and antagonists

1 reference

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5-HT2A receptors stimulate ACTH, corticosterone, oxytocin, renin, and prolactin release and activate hypothalamic CRF and oxytocin-expressing cells

1 reference

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Evidence that G(z)-proteins couple to hypothalamic 5-HT(1A) receptors in vivo.

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The role of 5-HT2A receptors in antipsychotic activity

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Chronic treatment with (+/-)DOI, a psychotomimetic 5-HT2 agonist, downregulates 5-HT2 receptors in rat brain

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The concept of selectivity in 5-HT receptor research

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5-Hydroxytryptamine2A (5-HT2A) receptor desensitization can occur without down-regulation

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Decreased frontal cortical serotonin2A receptors in schizophrenia.

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Paradoxical increase of 5-hydroxytryptamine2 receptors and 5-hydroxytryptamine2 receptor mRNA in cerebellar granule cells after persistent 5-hydroxytryptamine2 receptor stimulation.

1 reference

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Autoradiographic characterization of (+-)-1-(2,5-dimethoxy-4-[125I] iodophenyl)-2-aminopropane ([125I]DOI) binding to 5-HT2 and 5-HT1c receptors in rat brain.

1 reference

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Molecular pharmacological differences in the interaction of serotonin with 5-hydroxytryptamine1C and 5-hydroxytryptamine2 receptors

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Quantitative mapping shows that serotonin rather than dopamine receptor mRNA expressions are affected after repeated intermittent administration of MDMA in rat brain.

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Agonist-induced serotonin 2A receptor desensitization in the rat frontal cortex and hypothalamus

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Identification of two serine residues essential for agonist-induced 5-HT2A receptor desensitization

1 reference

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Chronic fluoxetine differentially affects 5-hydroxytryptamine (2A) receptor signaling in frontal cortex, oxytocin- and corticotropin-releasing factor-containing neurons in rat paraventricular nucleus

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Pharmacokinetics and brain distribution in non human primate of R(-)[123I]DOI, A 5HT(2A/2C) serotonin agonist

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Comparison of the potency of MDL 100,907 and SB 242084 in blocking the serotonin (5-HT)(2) receptor agonist-induced increases in rat serum corticosterone concentrations: evidence for 5-HT(2A) receptor mediation of the HPA axis

1 reference

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Characterization of the functional heterologous desensitization of hypothalamic 5-HT(1A) receptors after 5-HT(2A) receptor activation.

1 reference

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Ovarian steroid effects on serotonin 1A, 2A and 2C receptor mRNA in macaque hypothalamus.

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A desensitization of hypothalamic 5-HT1A receptors by repeated injections of paroxetine: reduction in the levels of G(i) and G(o) proteins and neuroendocrine responses, but not in the density of 5-HT1A receptors.

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Chronic mianserin treatment decreases 5-HT2 receptor binding without altering 5-HT2 receptor mRNA levels.

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1 reference

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based on heuristic

inferred from PubMed ID database lookup

Comparative localization of serotonin1A, 1C, and2 receptor subtype mRNAs in rat brain

1 reference

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based on heuristic

inferred from PubMed ID database lookup

Chronic fluoxetine or desmethylimipramine treatment alters 5-HT2 receptor mediated c-fos gene expression

1 reference

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1 reference

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1 reference

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based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.NEUROPHARM.2008.06.001

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Europe PubMed Central

17 August 2017

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Europe PubMed Central

17 August 2017

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Europe PubMed Central

17 August 2017

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