Allosteric antagonists of the muscarinic acetylcholine receptor (Q37204922)

18 August 2017

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title

Allosteric antagonists of the muscarinic acetylcholine receptor (English)

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18 August 2017

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

author name string

N. H. Lee

1

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1859442

11 December 2022

E. E. el-Fakahany

2

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1859442

11 December 2022

language of work or name

English

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publication date

1 July 1991

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18 August 2017

5 July 1991

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National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=1859442

full work available at URL

11 December 2022

https://api.elsevier.com/content/article/PII:0006295291907038?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

https://api.elsevier.com/content/article/PII:0006295291907038?httpAccept=text/plain

11 December 2022

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

11 December 2022

published in

Biochemical Pharmacology

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18 August 2017

volume

42

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18 August 2017

issue

2

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18 August 2017

page(s)

199-205

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Identification of a family of muscarinic acetylcholine receptor genes

18 August 2017

cites work

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A family of receptors coupled to guanine nucleotide regulatory proteins

11 December 2022

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Molecular biology of adrenergic and muscarinic cholinergic receptors. A perspective

11 December 2022

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Cloning, sequencing and expression of complementary DNA encoding the muscarinic acetylcholine receptor

11 December 2022

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Muscarinic receptor differentiation

11 December 2022

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ON THE NATURE OF ALLOSTERIC TRANSITIONS: A PLAUSIBLE MODEL

11 December 2022

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Comparison of Experimental Binding Data and Theoretical Models in Proteins Containing Subunits*

11 December 2022

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Pirenzepine distinguishes between different subclasses of muscarinic receptors

11 December 2022

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Modification of the binding properties of muscarinic receptors by gallamine

11 December 2022

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Some quantitative uses of drug antagonists

11 December 2022

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The Uptake of Atropine and Related Drugs by Intestinal Smooth Muscle of the Guinea-Pig in Relation to Acetylcholine Receptors

11 December 2022

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The inhibitory effect of gallamine on muscarinic receptors

11 December 2022

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Heterogeneity of binding sites on cardiac muscarinic receptors induced by the neuromuscular blocking agents gallamine and pancuronium

11 December 2022

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Stabilization of antagonist binding to cardiac muscarinic acetylcholine receptors by gallamine and other neuromuscular blocking drugs

11 December 2022

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Effects of d-tubocurarine on rat cardiac muscarinic receptors: a comparison with gallamine

11 December 2022

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The interaction of pancuronium with cardiac and ileal muscarinic receptors

11 December 2022

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The interaction of nicotinic receptor antagonists at muscarinic receptors.

11 December 2022

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Binding and functional characterization of the cardioselective muscarinic antagonist methoctramine

11 December 2022

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Allosteric interactions of three muscarine antagonists at bovine tracheal smooth muscle and cardiac M2 receptors

11 December 2022

29

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The allosteric binding profile of himbacine: a comparison with other cardioselective muscarinic antagonists

11 December 2022

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Characterization of the antimuscarinic effect of heptane-1,7-bis-(dimethyl-3'-phthalimidopropyl ammonium bromide).

11 December 2022

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The interaction of hexamethonium with muscarinic receptor subtypes in vitro

11 December 2022

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Inhibitory effects of quinidine on rat heart muscarinic receptors.

11 December 2022

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Interactions of quinidine and lidocaine with rat brain and heart muscarinic receptors

11 December 2022

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Bretylium tosylate binds preferentially to muscarinic receptors labelled with [3H]oxotremorine M (SH or 'high affinity' receptors) in rat heart and brain cortex

11 December 2022

35

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Interaction of DPI 201-106 with cardiac muscarinic receptors

11 December 2022

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Potassium channel blockers differentially affect carbachol and (-)-N6-phenylisopropyladenosine on guinea-pig atria

11 December 2022

37

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Effects of verapamil on the binding properties of rat heart muscarinic receptors: evidence for an allosteric site

11 December 2022

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Verapamil interaction with the muscarinic receptor: stereoselectivity at two sites

11 December 2022

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Gallamine exerts biphasic allosteric effects at muscarinic receptors

11 December 2022

40

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Characterization of guinea-pig cardiac muscarinic receptors by radioligand dissociation kinetics

11 December 2022

41

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The effect of McN-A-343 on muscarinic receptors in the cerebral cortex and heart

11 December 2022

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Myocardial muscarinic acetylcholine receptor: choline and tris unmask heterogeneity of antagonist binding sites.

11 December 2022

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Obligatory role of a Tris/choline allosteric site in guanine nucleotide regulation of [3H]-L-QNB binding to muscarinic acetylcholine receptors

11 December 2022

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Comparative binding studies with cholinergic ligands and histrionicotoxin at muscarinic receptors of neural cell lines

11 December 2022

45

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Allosteric effect of gallamine on muscarinic cholinergic receptor binding: influence of guanine nucleotides and conformational state

11 December 2022

46

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In vitro effects of gallamine on dissociation kinetics of (3H)N-methylscopolamine and (3H)pirenzepine from rat brain muscarinic receptors

11 December 2022

47

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Mixed competitive and allosteric antagonism by gallamine of muscarinic receptor-mediated second messenger responses in N1E-115 neuroblastoma cells.

11 December 2022

48

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Possible allosteric interaction of 4-aminopyridine with rat brain muscarinic acetylcholine receptors

11 December 2022

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Effects of verapamil on the binding characteristics of muscarinic receptor subtypes

11 December 2022

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Secoverine is a non-selective muscarinic antagonist on rat heart and brain receptors

11 December 2022

51

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Allosteric interactions between muscarinic agonist binding sites and effector sites demonstrated by the use of bisquaternary pyridinium oximes

11 December 2022

53

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The differential loss of [3H]pirenzepine vs [3H] (-) quinuclidinylbenzilate binding to soluble rat brain muscarinic receptors indicates that pirenzepine binds to an allosteric state of the muscarinic receptor

11 December 2022

54

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Multiple in vitro interactions with and differential in vivo regulation of muscarinic receptor subtypes by tetrahydroaminoacridine

11 December 2022

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Different mechanisms of antagonism by methoctramine of two neuronal muscarinic receptor-mediated second messenger responses

11 December 2022

57

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Antimuscarinic action of methoctramine, a new cardioselective M-2 muscarinic receptor antagonist, alone and in combination with atropine and gallamine

11 December 2022

58

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The interaction of methoctramine and himbacine at atrial, smooth muscle and endothelial muscarinic receptors in vitro

11 December 2022

59

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Competitive and non-competitive antagonism exhibited by 'selective' antagonists at atrial and ileal muscarinic receptor subtypes

11 December 2022

60

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Pharmacologic discrimination between receptor heterogeneity and allosteric interaction: resultant analysis of gallamine and pirenzepine antagonism of muscarinic responses in rat trachea

11 December 2022

62

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Differential allosteric effects of 8-(N,N-diethylamino)octyl-3,4,5-trimethoxybenzoate-HCl (TMB-8) on muscarinic receptor subtypes

11 December 2022

64

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The pharmacology of Flaxedil, with observations on certain analogs

11 December 2022

65

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

The sympathomimetic effect of gallamine on the heart

11 December 2022

66

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Regional distribution of muscarinic receptors preferring gallamine in the rat brain

11 December 2022

68

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The interaction of hemicholinium-3 (HC-3) with cholinomimetics and atropine

11 December 2022

69

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Muscarinic receptor heterogeneity in rat central nervous system. II. Brain receptors labeled by [3H]oxotremorine-M correspond to heterogeneous M2 receptors with very high affinity for agonists

11 December 2022

70

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Competitive interaction of gallamine with multiple muscarinic receptors

11 December 2022

71

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Characterization of the interactions of gallamine with muscarinic receptors from brain

11 December 2022

72

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Effects of gallamine triethiodide on membrane currents in amphibian and mammalian peripheral nerve

11 December 2022

76

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

GTP-binding proteins couple cardiac muscarinic receptors to a K channel.

11 December 2022

79

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Uncoupling of cardiac muscarinic and beta-adrenergic receptors from ion channels by a guanine nucleotide analogue

11 December 2022

80

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Polymethylene tetraamines as muscarinic receptor probes

11 December 2022

83

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https://api.crossref.org/works/10.1016/0006-2952(91)90703-8

Reduction of muscarinic acetylcholine receptor number and affinity by an endogenous substance

11 December 2022

84

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Endogenous inhibitor of ligand binding to the muscarinic acetylcholine receptor

11 December 2022

85

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11 December 2022

Identifiers

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18 August 2017

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