Netazepide, a gastrin/CCK2 receptor antagonist, causes dose-dependent, persistent inhibition of the responses to pentagastrin in healthy subjects. (Q37369301)

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English	Netazepide, a gastrin/CCK2 receptor antagonist, causes dose-dependent, persistent inhibition of the responses to pentagastrin in healthy subjects.	scientific article

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24 February 2020

Netazepide, a gastrin/CCK2 receptor antagonist, causes dose-dependent, persistent inhibition of the responses to pentagastrin in healthy subjects (English)

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24 February 2020

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24 February 2020

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Steve Warrington

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24 February 2020

James Black

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1 November 2013

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24 February 2020

British Journal of Clinical Pharmacology

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24 February 2020

689-698

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24 February 2020

Effect of repeated doses of netazepide, a gastrin receptor antagonist, omeprazole and placebo on 24 h gastric acidity and gastrin in healthy subjects

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6 September 2017

Guide to Receptors and Channels (GRAC), 5th edition

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6 September 2017

In vivo analysis of mouse gastrin gene regulation in enhanced GFP-BAC transgenic mice

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Reflections on some pilot trials of gastrin receptor blockade in pancreatic cancer

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6 September 2017

Control of gastric acid secretion in somatostatin receptor 2 deficient mice: shift from endocrine/paracrine to neurocrine pathways

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Genetically engineered mice: a new paradigm to study gastric physiology

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Attack and defence in the gastric epithelium - a delicate balance

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Review article: Pathogenesis and management of gastric carcinoid tumours.

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Genetic dissection of the signaling pathways that control gastric acid secretion

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Gastroduodenal mucus bicarbonate barrier: protection against acid and pepsin

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6 September 2017

Gastrin agonists and antagonists

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6 September 2017

Role of gastrin in the development of gastric mucosa, ECL cells and A-like cells in newborn and young rats

1 reference

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6 September 2017

Validation of a liquid chromatographic-tandem mass spectrometric method for the measurement of (R)-1-[2,3-dihydro-2-oxo-1-pivaloylmethyl-5-(2-pyridyl)-1H-1,4-benzodiazepin-3-yl]-3-(3-methylaminophenyl)urea (YF476) in human plasma

1 reference

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6 September 2017

Cellular expression of CCK-A and CCK-B/gastrin receptors in human gastric mucosa

1 reference

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6 September 2017

Mobilization of rat stomach ECL-cell histamine in response to short- or long-term treatment with omeprazole and/or YF 476 studied by gastric submucosal microdialysis in conscious rats

1 reference

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6 September 2017

The gastrins: their production and biological activities

1 reference

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6 September 2017

24-h recording of intragastric pH: technical aspects and clinical relevance.

1 reference

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6 September 2017

A double-blind, placebo-controlled study of a CCK-B receptor antagonist, CI-988, in patients with generalized anxiety disorder

1 reference

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6 September 2017

Gastric bicarbonate secretion in humans. Effect of pentagastrin, bethanechol, and 11,16,16-trimethyl prostaglandin E2

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

6 September 2017

Gastric acid secretion rate and buffer content of the stomach after eating. Results in normal subjects and in patients with duodenal ulcer

1 reference

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6 September 2017

Carbonic anhydrase in the normal rat stomach and duodenum and after treatment with omeprazole and ranitidine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

6 September 2017

Relationship between undissociated acidity of gastric juice and gastric protein secreted in response to graded doses of pentagastrin in duodenal ulcer patients

1 reference

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6 September 2017

Gastrin activates paracrine networks leading to induction of PAI-2 via MAZ and ASC-1.

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14 September 2017

Gastrin regulates the TFF2 promoter through gastrin-responsive cis-acting elements and multiple signaling pathways.

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14 September 2017

Measurement of gastric bicarbonate secretion in the human stomach: different methods produce discordant results

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28 September 2017

Effects of YF476, a potent and selective gastrin/cholecystokinin-B receptor antagonist, on gastric acid secretion in beagle dogs with gastric fistula.

1 reference

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26 June 2018

YF476 is a new potent and selective gastrin/cholecystokinin-B receptor antagonist in vitro and in vivo

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

26 June 2018

(3R)-N-(1-(tert-butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H-1,4-benzodiazepin-3-yl)-N'-(3-(methylamino)phenyl)urea (YF476): a potent and orally active gastrin/CCK-B antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

26 June 2018

Does antral distension inhibit gastric acid secretion or stimulate bicarbonate secretion in 'healthy' subjects?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

26 June 2018

Vagal stimulation of human gastric bicarbonate secretion.

1 reference

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26 June 2018

Vagal cholinergic control of gastric alkaline secretion in normal subjects and duodenal ulcer patients

1 reference

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26 June 2018

Treatment of gastric carcinoids type 1 with the gastrin receptor antagonist netazepide (YF476) results in regression of tumours and normalisation of serum chromogranin A.

1 reference

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2 September 2018

Single oral doses of netazepide (YF476), a gastrin receptor antagonist, cause dose-dependent, sustained increases in gastric pH compared with placebo and ranitidine in healthy subjects.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Dyspeptic symptom development after discontinuation of a proton pump inhibitor: a double-blind placebo-controlled trial

1 reference

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2 September 2018

Complexity of gastric acid secretion revealed by targeted gene disruption in mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

The CCK(2) receptor antagonist, YF476, inhibits Mastomys ECL cell hyperplasia and gastric carcinoid tumor development

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Proton-pump inhibitor therapy induces acid-related symptoms in healthy volunteers after withdrawal of therapy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Gastric acid secretion in cholecystokinin-1 receptor, -2 receptor, and -1, -2 receptor gene knockout mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Synergistic inhibitory effects of gastrin and histamine receptor antagonists on Helicobacter-induced gastric cancer.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Spontaneous ECL cell carcinomas in cotton rats: natural course and prevention by a gastrin receptor antagonist.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Effect of long-term, continuous versus alternate-day omeprazole therapy on serum gastrin in patients treated for reflux esophagitis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

Long-lasting cholecystokinin(2) receptor blockade after a single subcutaneous injection of YF476 or YM022.

1 reference

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2 September 2018

The gastrin-receptor antagonist L-365,260 inhibits stimulated acid secretion in humans

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3853528

2 September 2018

A demonstration of bicarbonate production by the normal human stomach in vivo

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

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Effects of spiroglumide, a gastrin receptor antagonist, on acid secretion in humans

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

based on heuristic

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Positioning of Subject and of Nasogastric Tube during a Gastric Secretion Study

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

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A placebo-controlled trial of L-365,260, a CCKB antagonist, in panic disorder

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Electrolytes in gastric juice of man. I. A statistical analysis of calcium and inorganic phosphorus before and after subcutaneous injection of large doses of histamine

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

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inferred from PubMed ID database lookup

Gastric H+ and HCO3- secretion in response to sham feeding in humans

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

based on heuristic

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Gastrin-induced apoptosis contributes to carcinogenesis in the stomach

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

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The buffer substances of the gastric juice, and their relation to gastric mucus

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

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Undissociated acidity of human gastric juice. Measurement and relationship to protein buffers

1 reference

https://pubmed.ncbi.nlm.nih.gov/23432534

12 December 2020

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Tolerance during 8 days of high-dose H2-blockade: placebo-controlled studies of 24-hour acidity and gastrin

1 reference

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12 December 2020

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Evaluation of three novel cholecystokinin-B/gastrin receptor antagonists: a study of their effects on rat stomach enterochromaffin-like cell activity

1 reference

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12 December 2020

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inferred from PubMed ID database lookup

Transcriptional regulation of the human trefoil factor, TFF1, by gastrin

1 reference

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12 December 2020

based on heuristic

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Problems with the interpretation of gastric pH measurement

1 reference

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12 December 2020

based on heuristic

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Increased risk of fundic gland polyps during long-term proton pump inhibitor therapy

1 reference

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Identifiers

10.1111/BCP.12099

1 reference

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24 February 2020

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23432534%20AND%20SRC:MED&resulttype=core&format=json

24 February 2020

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23432534%20AND%20SRC:MED&resulttype=core&format=json

24 February 2020

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