The beta-D-glucose scaffold as a beta-turn mimetic (Q37394232)

20 August 2017

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title

The beta-D-glucose scaffold as a beta-turn mimetic (English)

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20 August 2017

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Ralph F Hirschmann

1

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20 August 2017

K C Nicolaou

2

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20 August 2017

Angie R Angeles

3

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20 August 2017

Jason S Chen

4

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20 August 2017

Amos B Smith

5

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20 August 2017

language of work or name

English

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publication date

1 October 2009

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Accounts of Chemical Research

20 August 2017

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20 August 2017

42

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20 August 2017

10

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20 August 2017

1511-1520

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Enzyme dynamics during catalysis

20 August 2017

1 reference

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Cellular biology of somatostatin receptors

6 September 2017

1 reference

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Crystal structure of rhodopsin: A G protein-coupled receptor

6 September 2017

1 reference

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Comprehensive survey of combinatorial library synthesis: 1998.

6 September 2017

1 reference

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New 4-point pharmacophore method for molecular similarity and diversity applications: overview of the method and applications, including a novel approach to the design of combinatorial libraries containing privileged substructures

6 September 2017

1 reference

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Rational design and combinatorial evaluation of enzyme inhibitor scaffolds: identification of novel inhibitors of matrix metalloproteinases

6 September 2017

1 reference

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RECAP--retrosynthetic combinatorial analysis procedure: a powerful new technique for identifying privileged molecular fragments with useful applications in combinatorial chemistry

6 September 2017

1 reference

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CLUSTAL W: improving the sensitivity of progressive multiple sequence alignment through sequence weighting, position-specific gap penalties and weight matrix choice

6 September 2017

1 reference

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Proposed conformation of oxytocin in solution

6 September 2017

1 reference

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Conformationally restricted analogs of somatostatin with high mu-opiate receptor specificity

6 September 2017

1 reference

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Cloning and functional characterization of a family of human and mouse somatostatin receptors expressed in brain, gastrointestinal tract, and kidney

6 September 2017

1 reference

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Identification of two related pentapeptides from the brain with potent opiate agonist activity

6 September 2017

1 reference

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Conformationally restricted bicyclic analogs of somatostatin

6 September 2017

1 reference

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Biologic and immunologic activities and applications of somatostatin analogs

6 September 2017

1 reference

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Modulation of receptor and receptor subtype affinities using diastereomeric and enantiomeric monosaccharide scaffolds as a means to structural and biological diversity. A new route to ether synthesis

14 September 2017

1 reference

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The properties of known drugs. 1. Molecular frameworks

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2764824

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2764824

Molecular pharmacology of somatostatin receptor subtypes

28 September 2017

1 reference

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Approaches to vasodilating/.beta.-adrenergic blocking agents: examples of the dihydrolutidine type

26 June 2018

1 reference

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Topochemical investigations of peptide systems.

26 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2764824

Isolation of somatostatin (a somatotropin release inhibiting factor) of ovine hypothalamic origin

26 June 2018

1 reference

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Molecular forces governing non-electrolyte permeation through cell membranes.

26 June 2018

1 reference

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D-Trp8-somatostatin: An analog of somatostatin more potent than the native molecule

26 June 2018

1 reference

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(Acylaryloxy)acetic acid diuretics. 1. (2-Alkyl- and 2,2-dialkyl-1-oxo-5-indanyloxy)acetic acids

26 June 2018

1 reference

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Highly active cyclic and bicyclic somatostatin analogues of reduced ring size

26 June 2018

1 reference

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Effects of Heterocyclic Aromatic Substituents on Binding Affinities at Two Distinct Sites of Somatostatin Receptors. Correlation with the Electrostatic Potential of the Substituents

26 June 2018

1 reference

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G-Protein coupled receptors: models, mutagenesis, and drug design

2 September 2018

1 reference

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SMS 201–995: A very potent and selective octapeptide analogue of somatostatin with prolonged action

2 September 2018

1 reference

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Conformation of the LL and LD hairpin bends with internal hydrogen bonds in proteins and peptides

2 September 2018

1 reference

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Synthesis of a substance P antagonist with a somatostatin scaffold: factors affecting agonism/antagonism at GPCRs and the role of pseudosymmetry

2 September 2018

1 reference

12 December 2020

On the low energy solution conformation of somatostatin

1 reference

12 December 2020

A potent cyclic hexapeptide analogue of somatostatin

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12 December 2020

A super active cyclic hexapeptide analog of somatostatin

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12 December 2020

Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

1 reference

12 December 2020

Somatostatin receptors

1 reference

12 December 2020

Peptide Mimetics of Thyrotropin-Releasing Hormone Based on a Cyclohexane Framework: Design, Synthesis, and Cognition-Enhancing Properties

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12 December 2020

Molecular biology of somatostatin receptors

1 reference

12 December 2020

Synthesis of potent cyclic hexapeptide NK-1 antagonists. Use of a minilibrary in transforming a peptidal somatostatin receptor ligand into an NK-1 receptor ligand via a polyvalent peptidomimetic

1 reference

12 December 2020

Identifiers

DOI

10.1021/AR900020X

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20 August 2017

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20 August 2017

PubMed publication ID

19624154

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