Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC. (Q37396399)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18603240%20AND%20SRC:MED&resulttype=core&format=json

10 January 2020

title

Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18603240%20AND%20SRC:MED&resulttype=core&format=json

10 January 2020

3

1 reference

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10 January 2020

Gunnar Schulte

5

1 reference

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10 January 2020

author name string

Frank Brand

1

1 reference

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10 January 2020

Athena M Klutz

2

1 reference

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10 January 2020

Bertil B Fredholm

4

1 reference

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10 January 2020

language of work or name

English

0 references

publication date

4 July 2008

1 reference

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European Journal of Pharmacology

10 January 2020

published in

1 reference

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10 January 2020

volume

590

1 reference

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10 January 2020

issue

1-3

1 reference

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10 January 2020

page(s)

36-42

1 reference

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G protein-coupled receptor trafficking in health and disease: lessons learned to prepare for therapeutic mutant rescue in vivo

10 January 2020

cites work

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Clathrin-dependent mechanisms of G protein-coupled receptor endocytosis

6 September 2017

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Beta-arrestins and cell signaling

6 September 2017

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6 September 2017

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The ubiquitin-specific protease Usp4 regulates the cell surface level of the A2A receptor

6 September 2017

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6 September 2017

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"Reversine" and its 2-substituted adenine derivatives as potent and selective A3 adenosine receptor antagonists

6 September 2017

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2-Substituted adenosine derivatives: affinity and efficacy at four subtypes of human adenosine receptors

6 September 2017

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Differential kinetic and spatial patterns of beta-arrestin and G protein-mediated ERK activation by the angiotensin II receptor

6 September 2017

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Quantitative analysis of the formation and diffusion of A1-adenosine receptor-antagonist complexes in single living cells

6 September 2017

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Fluorescent ligands, antibodies, and proteins for the study of receptors

6 September 2017

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The adenosine A2A receptor interacts with the actin-binding protein alpha-actinin

6 September 2017

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Signalling from adenosine receptors to mitogen-activated protein kinases

6 September 2017

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Pharmacology of adenosine A2A receptors and therapeutic applications

6 September 2017

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Subtype-specific regulation of receptor internalization and recycling by the carboxyl-terminal domains of the human A1 and rat A3 adenosine receptors: consequences for agonist-stimulated translocation of arrestin3

6 September 2017

1 reference

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Coaggregation, cointernalization, and codesensitization of adenosine A2A receptors and dopamine D2 receptors

6 September 2017

1 reference

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International Union of Pharmacology. XXV. Nomenclature and classification of adenosine receptors

6 September 2017

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Role of endocytosis in the activation of the extracellular signal-regulated kinase cascade by sequestering and nonsequestering G protein-coupled receptors.

6 September 2017

1 reference

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Enhanced expression of G protein-coupled receptor kinase 2 selectively increases the sensitivity of A2A adenosine receptors to agonist-induced desensitization

6 September 2017

1 reference

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Clathrin-mediated endocytosis of the beta-adrenergic receptor is regulated by phosphorylation/dephosphorylation of beta-arrestin1

6 September 2017

1 reference

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Aggressiveness, hypoalgesia and high blood pressure in mice lacking the adenosine A2a receptor

6 September 2017

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125I-4-(2-[7-amino-2-[2-furyl][1,2,4]triazolo[2,3-a][1,3,5] triazin-5-yl-amino]ethyl)phenol, a high affinity antagonist radioligand selective for the A2a adenosine receptor

6 September 2017

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The in vitro pharmacology of ZM 241385, a potent, non‐xanthine, A2a selective adenosine receptor antagonist

6 September 2017

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Agonist derived molecular probes for A2 adenosine receptors

6 September 2017

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Molecular characterization of a human brain adenosine A2 receptor

6 September 2017

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A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase

6 September 2017

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Tumor necrosis factor-alpha prevents desensitization of Galphas-coupled receptors by regulating GRK2 association with the plasma membrane

6 September 2017

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Agonist-receptor-arrestin, an alternative ternary complex with high agonist affinity.

14 September 2017

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Desensitization of the canine A2a adenosine receptor: delineation of multiple processes.

28 September 2017

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A FlAsH-based FRET approach to determine G protein-coupled receptor activation in living cells

28 September 2017

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Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.

26 June 2018

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Hypertonic media inhibit receptor-mediated endocytosis by blocking clathrin-coated pit formation

26 June 2018

1 reference

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New fluorescent adenosine A1-receptor agonists that allow quantification of ligand-receptor interactions in microdomains of single living cells.

26 June 2018

1 reference

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The G(s)-coupled adenosine A(2B) receptor recruits divergent pathways to regulate ERK1/2 and p38.

2 September 2018

1 reference

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Rapid agonist-induced desensitization and internalization of the A(2B) adenosine receptor is mediated by a serine residue close to the COOH terminus

2 September 2018

1 reference

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Endosome fusion in living cells overexpressing GFP-rab5.

2 September 2018

1 reference

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Reciprocal interactions between adenosine A2A and dopamine D2 receptors in Chinese hamster ovary cells co-transfected with the two receptors

2 September 2018

1 reference

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The effect of inhibitors of receptor internalization on the desensitization and resensitization of three Gs-coupled receptor responses

2 September 2018

1 reference

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A dominant negative mutant of the G protein-coupled receptor kinase 2 selectively attenuates adenosine A2 receptor desensitization.

2 September 2018

1 reference

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Identification of an A2a adenosine receptor domain specifically responsible for mediating short-term desensitization

2 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18603240

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Human adenosine A(1), A(2A), A(2B), and A(3) receptors expressed in Chinese hamster ovary cells all mediate the phosphorylation of extracellular-regulated kinase 1/2

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/18603240

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.EJPHAR.2008.05.036

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18603240%20AND%20SRC:MED&resulttype=core&format=json

10 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18603240%20AND%20SRC:MED&resulttype=core&format=json

10 January 2020

PubMed publication ID

18603240

1 reference