Characterization of putative GRP- and NMB-receptor antagonist's interaction with human receptors. (Q37398035)

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28 January 2020

title

Characterization of putative GRP- and NMB-receptor antagonist's interaction with human receptors (English)

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28 January 2020

author name string

Samuel A Mantey

2

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28 January 2020

Tapas K Pradhan

3

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28 January 2020

Veronica Sancho

4

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28 January 2020

Terry W Moody

5

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28 January 2020

Robert T Jensen

7

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28 January 2020

publication date

20 May 2009

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28 January 2020

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20 August 2017

30

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28 January 2020

issue

8

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28 January 2020

page(s)

1473-1486

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Regulation and signaling of human bombesin receptors and their biological effects

28 January 2020

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BRS-3: a novel bombesin receptor subtype selectively expressed in testis and lung carcinoma cells

6 September 2017

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Expression and characterization of cloned human bombesin receptors

6 September 2017

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Differential activation of human gastrin-releasing peptide receptor-mediated responses by bombesin analogs.

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14 September 2017

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28 September 2017

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Neuromedin B receptors retain functional expression when transfected into BALB 3T3 fibroblasts: analysis of binding, kinetics, stoichiometry, modulation by guanine nucleotide-binding proteins, and signal transduction and comparison with natively exp

28 September 2017

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26 June 2018

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26 June 2018

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Characterization of bombesin receptors using a novel, potent, radiolabeled antagonist that distinguishes bombesin receptor subtypes

26 June 2018

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Peptide structural requirements for antagonism differ between the two mammalian bombesin receptor subtypes

26 June 2018

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A synthetic peptide that is a bombesin receptor antagonist

26 June 2018

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Neuromedin B receptor in esophagus: evidence for subtypes of bombesin receptors

26 June 2018

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Effect of substitutions in position 12 of bombesin on antagonist activity

26 June 2018

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Short-chain pseudopeptide bombesin receptor antagonists with enhanced binding affinities for pancreatic acinar and Swiss 3T3 cells display strong antimitotic activity

26 June 2018

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Characterization of ability of various substance P antagonists to inhibit action of bombesin

26 June 2018

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26 June 2018

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26 June 2018

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26 June 2018

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26 June 2018

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26 June 2018

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26 June 2018

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Effect of the bombesin receptor blockers [Leu13,ψCH2NH-Leu14]bombesin and N-pivaloyl GRP(20–25) alkylamide (L 686,095-001C002) on basal and neuromedin C-stimulated PRL and GH release in pituitary cell aggregates

26 June 2018

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Distinct distributions of two bombesin receptor subtypes in the rat central nervous system

26 June 2018

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Neuromedin B binds with high affinity, elevates cytosolic calcium and stimulates the growth of small-cell lung cancer cell lines

26 June 2018

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Development of a potent bombesin receptor antagonist with prolonged in vivo inhibitory activity on bombesin-stimulated amylase and protein release in the rat

26 June 2018

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Development of high affinity camptothecin-bombesin conjugates that have targeted cytotoxicity for bombesin receptor-containing tumor cells

10 July 2018

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Gastrin-releasing peptide receptor-induced internalization, down-regulation, desensitization, and growth: possible role for cyclic AMP.

2 September 2018

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Potent bombesin receptor antagonists distinguish receptor subtypes

2 September 2018

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12 December 2020

Characterization of functional receptors for gastrointestinal hormones on human colon cancer cells

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12 December 2020

Effect of [D-Phe6] bombesin (6-13) methylester, a bombesin receptor antagonist, towards bombesin-induced contractions in the guinea-pig and rat isolated urinary bladder

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12 December 2020

Species differences of bombesin analog interactions with GRP-R define the choice of animal models in the development of GRP-R-targeting drugs

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12 December 2020

Bombesin receptor subtypes in human cancers: detection with the universal radioligand (125)I-[D-TYR(6), beta-ALA(11), PHE(13), NLE(14)] bombesin(6-14)

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12 December 2020

Partial agonist activity of the bombesin-receptor antagonist [Leu14-psi-CH2-NH-Leu13]-bombesin in frog peptic cells

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12 December 2020

10.1016/J.PEPTIDES.2009.05.007

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19463875%20AND%20SRC:MED&resulttype=core&format=json

28 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:19463875%20AND%20SRC:MED&resulttype=core&format=json

28 January 2020

PubMed publication ID

19463875

1 reference