Complete differentiation between enkephalinase and angiotensin-converting enzyme inhibition by retro-thiorphan (Q37613022)

21 August 2017

Complete differentiation between enkephalinase and angiotensin-converting enzyme inhibition by retro-thiorphan (English)

1 reference

21 August 2017

B. P. Roques

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

22 September 2023

E. Lucas-Soroca

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

22 September 2023

P. Chaillet

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

22 September 2023

J. Costentin

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

22 September 2023

M. C. Fournié-Zaluski

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

22 September 2023

language of work or name

English

0 references

publication date

1 June 1983

1 reference

PMCID

394003

full work available at URL

21 August 2017

https://europepmc.org/articles/pmc394003?pdf=render

file format

Portable Document Format

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

https://europepmc.org/articles/PMC394003

22 September 2023

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

https://europepmc.org/articles/PMC394003?pdf=render

22 September 2023

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A6304695

https://pnas.org/doi/pdf/10.1073/pnas.80.11.3178

22 September 2023

1 reference

Crossref

DOI

10.1073/PNAS.80.11.3178

https://api.crossref.org/works/10.1073/PNAS.80.11.3178

Proceedings of the National Academy of Sciences of the United States of America

22 September 2023

published in

1 reference

21 August 2017

80

1 reference

21 August 2017

11

1 reference

21 August 2017

3178-3182

1 reference

Binding of ligands to the active site of carboxypeptidase A

21 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

The purification and specificity of a neutral endopeptidase from rabbit kidney brush border

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Identification of two related pentapeptides from the brain with potent opiate agonist activity

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Morphine-like peptides in mammalian brain: isolation, structure elucidation, and interactions with the opiate receptor

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Design of Specific Inhibitors of Angiotensin-Converting Enzyme: New Class of Orally Active Antihypertensive Agents

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

In vitro degradation of enkephalin: evidence for cleavage at the Gly-Phe bond

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Enzymes of the Renin-Angiotensin System and their Inhibitors

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Two distinct enkephalinases: Solubilization, partial purification and separation from angiotensin converting enzyme

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Co-identity of brain angiotensin converting enzyme with a membrane bound dipeptidyl carboxypeptidase inactivating Met-enkephalin

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

High-affinity enkephalin-degrading peptidase in brain is increased after morphine

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Pharmacological effects produced by intracerebral injection of drugs in the conscious mouse

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Structure of a mercaptan-thermolysin complex illustrates mode of inhibition of zinc proteases by substrate-analogue mercaptans

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Phosphoryl-Leu-Phe: a potent inhibitor of the degradation of enkephalin by enkephalinase

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Degradation of exogenous enkephalin in the guinea-pig ileum: relative importance of aminopeptidase, enkephalinase and angiotensin converting enzyme activity

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Mode of deactivation of the enkephalins by rat and human plasma and rat brain homogenates

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Inhibitory potency of various peptides on enkephalinase activity from mouse striatum

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Partially modified retro-inverso-enkephalinamides: topochemical long-acting analogs in vitro and in vivo

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Design of potent and specific inhibitors of carboxypeptidases A and B

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Multiple molecular forms of rat brain enkephalinase.

25 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

Enkephalin dipeptidyl carboxypeptidase (enkephalinase) activity: selective radioassay, properties, and regional distribution in human brain.

1 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

New carboxyalkyl inhibitors of brain enkephalinase: synthesis, biological activity, and analgesic properties.

1 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=394003

A crystallographic study of the complex of phosphoramidon with thermolysin. A model for the presumed catalytic transition state and for the binding of extended substances

1 September 2018

1 reference

12 December 2020

Hydrolysis of enkephalin by cultured human endothelial cells and by purified peptidyl dipeptidase

1 reference

12 December 2020

The enkephalinase inhibitor thiorphan shows antinociceptive activity in mice

1 reference

12 December 2020

Rational design of enkephalinase inhibitors: substrate specificity of enkephalinase studied from inhibitory potency of various dipeptides

1 reference

12 December 2020

Purification and specificity of a membrane-bound metalloendopeptidase from bovine pituitaries

1 reference

12 December 2020

Membrane bound pituitary metalloendopeptidase: apparent identity to enkephalinase

1 reference

12 December 2020

Effects of thiorphan on the antinociceptive actions of intrathecal [D-Ala2,Met5] enkephalin

1 reference

12 December 2020

Properties of "enkephalinase" from rat kidney: comparison of dipeptidyl-carboxypeptidase and endopeptidase activities

1 reference

12 December 2020

Thiorphan potentiation of stress-induced analgesia in the mouse

1 reference

12 December 2020

Potentiation of [D-ala2]enkephalinamide analgesia in rats by thiorphan

1 reference

12 December 2020

A method for evaluating both non-narcotic and narcotic analgesics

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.80.11.3178

1 reference

21 August 2017

0 references

1 reference

21 August 2017

1 reference

PMCID

394003