Synthesis and binding affinities of fluoroalkylated raloxifenes (Q38519804)

3 September 2017

title

Synthesis and binding affinities of fluoroalkylated raloxifenes (English)

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3 September 2017

Kyo Chul Lee

1

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3 September 2017

Byung Seok Moon

2

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3 September 2017

Jae Hak Lee

3

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3 September 2017

Kyoo-Hyun Chung

4

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3 September 2017

John A Katzenellenbogen

5

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3 September 2017

Dae Yoon Chi

6

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3 September 2017

language of work or name

English

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publication date

1 August 2003

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Bioorganic & Medicinal Chemistry

3 September 2017

published in

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3 September 2017

volume

11

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3 September 2017

issue

17

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3 September 2017

page(s)

3649-3658

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Synthesis and biological evaluation of 4-(hydroxyalkyl)estradiols and related compounds

3 September 2017

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Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: evidence that an open pocket conformation is required for ligand interaction.

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Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta

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Synthesis, radiolabeling and tissue distribution of 11 beta-fluoroalkyl- and 11 beta-fluoroalkoxy-substituted estrogens: target tissue uptake selectivity and defluorination of a homologous series of fluorine-18-labeled estrogens

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7 January 2021

10.1016/S0968-0896(03)00362-6

Identifiers

DOI

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3 September 2017

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