Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes. (Q39041277)

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5 April 2020

title

Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes (English)

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5 April 2020

2

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5 April 2020

Lyn H. Jones

6

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5 April 2020

Qian Zhao

1

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5 April 2020

Jack Taunton

8

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5 April 2020

author name string

Xiaobo Wan

3

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5 April 2020

Ketan S Gajiwala

4

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5 April 2020

John C Kath

5

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5 April 2020

Alma L Burlingame

7

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5 April 2020

language of work or name

English

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publication date

4 January 2017

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Journal of the American Chemical Society

5 April 2020

published in

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5 April 2020

volume

139

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5 April 2020

issue

2

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5 April 2020

page(s)

680-685

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Sulfonyl fluorides as privileged warheads in chemical biology

5 April 2020

cites work

1 reference

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The promise and peril of chemical probes

30 June 2018

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New affinity probe targeting VEGF receptors for kinase inhibitor selectivity profiling by chemical proteomics.

30 June 2018

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Characterization of a chemical affinity probe targeting Akt kinases

30 June 2018

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Characterization of the novel broad-spectrum kinase inhibitor CTx-0294885 as an affinity reagent for mass spectrometry-based kinome profiling.

30 June 2018

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Aromatic Sulfonyl Fluorides Covalently Kinetically Stabilize Transthyretin to Prevent Amyloidogenesis while Affording a Fluorescent Conjugate

30 June 2018

1 reference

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Affinity profiling of the cellular kinome for the nucleotide cofactors ATP, ADP, and GTP.

30 June 2018

1 reference

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Selective targeting of distinct active site nucleophiles by irreversible SRC-family kinase inhibitors

30 June 2018

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Affinity-Based Probes Based on Type II Kinase Inhibitors

30 June 2018

1 reference

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In situ kinase profiling reveals functionally relevant properties of native kinases

30 June 2018

1 reference

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Phase II study of dasatinib in patients with advanced non-small-cell lung cancer

30 June 2018

1 reference

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Tuning a Three-Component Reaction For Trapping Kinase Substrate Complexes

30 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5858558

A quantitative analysis of kinase inhibitor selectivity

30 June 2018

1 reference

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Dasatinib, a small-molecule protein tyrosine kinase inhibitor, inhibits T-cell activation and proliferation

30 June 2018

1 reference

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Quantitative chemical proteomics reveals mechanisms of action of clinical ABL kinase inhibitors

30 June 2018

1 reference

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Functional interrogation of the kinome using nucleotide acyl phosphates

30 June 2018

1 reference

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2-aminothiazole as a novel kinase inhibitor template. Structure-activity relationship studies toward the discovery of N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1- piperazinyl)]-2-methyl-4-pyrimidinyl]amino)]-1,3-thiazole-5-carboxamide (d

30 June 2018

1 reference

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A small molecule-kinase interaction map for clinical kinase inhibitors

30 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5858558

Affinity labeling of purine nucleotide sites in proteins

30 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5858558

Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.

30 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5858558

Current compound coverage of the kinome.

21 August 2018

1 reference

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Chemical proteomics with sulfonyl fluoride probes reveals selective labeling of functional tyrosines in glutathione transferases

21 August 2018

1 reference

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Cell-based proteome profiling of potential dasatinib targets by use of affinity-based probes.

21 August 2018

1 reference

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Lck is a key target of imatinib and dasatinib in T-cell activation

21 August 2018

1 reference

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Metabolism and disposition of dasatinib after oral administration to humans

21 August 2018

1 reference

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The Src/ABL kinase inhibitor dasatinib (BMS-354825) inhibits function of normal human T-lymphocytes in vitro

21 August 2018

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Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes

21 August 2018

1 reference

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A new chemical probe for quantitative proteomic profiling of fibroblast growth factor receptor and its inhibitors

2 December 2018

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Toward a pharmacophore for kinase frequent hitters

2 December 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/28051857

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JACS.6B08536

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28051857%20AND%20SRC:MED&resulttype=core&format=json

5 April 2020

1 reference

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5 April 2020

PubMed publication ID

28051857

1 reference