Rapid synthesis of new DNMT inhibitors derivatives of procainamide (Q39428367)

11 September 2017

title

Rapid synthesis of new DNMT inhibitors derivatives of procainamide (English)

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Dominique Guianvarc'h

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Olivier Lequin

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Thierry Drujon

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object named as

Thierry Drujon

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Alexandre Ceccaldi

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Paola B Arimondo

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Catherine Sénamaud-Beaufort

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object named as

Catherine Sénamaud-Beaufort

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Renata Jurkowska

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Ludovic Halby

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Christine Champion

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Sophie Ajjan

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William G Nelson

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Alain Guy

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Clotilde Ferroud

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publication date

14 December 2011

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volume

13

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issue

1

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page(s)

157-165

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CpG islands--'a rough guide'.

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cites work

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Procainamide is a specific inhibitor of DNA methyltransferase 1.

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Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1.

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Molecular basis of the targeting of topoisomerase II-mediated DNA cleavage by VP16 derivatives conjugated to triplex-forming oligonucleotides

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Targeting MDR1 gene: synthesis and cellular study of modified daunomycin-triplex-forming oligonucleotide conjugates able to inhibit gene expression in resistant cell lines.

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Design, synthesis, inhibitory activity, and binding mode study of novel DNA methyltransferase 1 inhibitors

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Synthesis and in vitro evaluation of biotinylated RG108: a high affinity compound for studying binding interactions with human DNA methyltransferases

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A detergent-based assay for the detection of promiscuous inhibitors

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Effect of detergent on "promiscuous" inhibitors

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Molecular modeling and molecular dynamics studies of hydralazine with human DNA methyltransferase 1.

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Structure and substrate recognition of the Escherichia coli DNA adenine methyltransferase

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Specificity of protein lysine methyltransferases and methods for detection of lysine methylation of non-histone proteins

21 January 2018

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Biotin-avidin microplate assay for the quantitative analysis of enzymatic methylation of DNA by DNA methyltransferases

21 January 2018

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Constrained (l-)-S-adenosyl-l-homocysteine (SAH) analogues as DNA methyltransferase inhibitors

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Structure of Dnmt3a bound to Dnmt3L suggests a model for de novo DNA methylation

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Identifiers

DOI

10.1002/CBIC.201100522

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11 September 2017

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