Discovery of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors (Q39782128)

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scientific article published on November 2009
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Discovery of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors
scientific article published on November 2009

    Statements

    Discovery of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors (English)
    Philip Jones
    Sergio Altamura
    Julia Boueres
    Federica Ferrigno
    Massimiliano Fonsi
    Claudia Giomini
    Stefania Lamartina
    Jesus M Ontoria
    Maria Vittoria Orsale
    Maria Cecilia Palumbi
    Silvia Pesci
    Giuseppe Roscilli
    Rita Scarpelli
    Michael Rowley
    1 November 2009
    7170-7185

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