Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity (Q39994950)

16 September 2017

title

Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity (English)

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6

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José Morais

2

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Bente Steffansen

object named as

Bente Steffansen

series ordinal

7

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Christophe Pannecouque

object named as

Christophe Pannecouque

series ordinal

5

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Erik De Clercq

object named as

Erik de Clercq

series ordinal

4

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publication date

1 June 2008

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16 September 2017

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volume

3

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issue

6

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16 September 2017

page(s)

970-978

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The efficacy of azidothymidine (AZT) in the treatment of patients with AIDS and AIDS-related complex. A double-blind, placebo-controlled trial

16 September 2017

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5'-Amino acid esters of antiviral nucleosides, acyclovir, and AZT are absorbed by the intestinal PEPT1 peptide transporter

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Synthesis and characterization of novel dipeptide ester prodrugs of acyclovir

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Amino acid ester prodrugs of the antiviral agent 2-bromo-5,6-dichloro-1-(beta-D-ribofuranosyl)benzimidazole as potential substrates of hPEPT1 transporter

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Conjugation of dipeptide to fluorescent dyes enhances its affinity for a dipeptide transporter (PEPT1) in human intestinal Caco-2 cells

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Identifiers

DOI

10.1002/CMDC.200800012

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16 September 2017

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