Assessment of stereoselectivity of trimethylphenylalanine analogues of delta-opioid [D-Pen(2),D-Pen(5)]-enkephalin. (Q40760933)

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7 November 2019

title

Assessment of stereoselectivity of trimethylphenylalanine analogues of delta-opioid [D-Pen(2),D-Pen(5)]-enkephalin (English)

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7 November 2019

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7

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7 November 2019

author name string

K A Witt

1

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7 November 2019

C A Slate

2

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7 November 2019

R D Egleton

3

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7 November 2019

J D Huber

4

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7 November 2019

H I Yamamura

5

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7 November 2019

V J Hruby

6

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7 November 2019

language of work or name

English

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publication date

1 July 2000

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Journal of Neurochemistry

7 November 2019

published in

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7 November 2019

volume

75

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7 November 2019

issue

1

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7 November 2019

page(s)

424-435

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Delivery of loperamide across the blood-brain barrier with polysorbate 80-coated polybutylcyanoacrylate nanoparticles.

7 November 2019

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Enhanced antinociception of the model opioid peptide [D-penicillamine] enkephalin by P-glycoprotein modulation

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Transport of the delta-opioid receptor agonist [D-penicillamine2,5] enkephalin across the blood-brain barrier involves transcytosis1.

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Metkephamid, a Systemically Active Analog of Methionine Enkephalin with Potent Opioid δ-Receptor Activity

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P-Glycoprotein on astrocyte foot processes of unfixed isolated human brain capillaries.

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A non-invasive system for delivering neural growth factors across the blood-brain barrier: a review

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Mode of deactivation of the enkephalins by rat and human plasma and rat brain homogenates

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Systemic analgesic activity and delta-opioid selectivity in [2,6-dimethyl-Tyr1,D-Pen2,D-Pen5]enkephalin

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Cyclic enkephalin analogues with exceptional potency and selectivity for delta-opioid receptors

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Identification of two related pentapeptides from the brain with potent opiate agonist activity

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Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides

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