GR94839, a kappa-opioid agonist with limited access to the central nervous system, has antinociceptive activity (Q42016685)

15 October 2017

GR94839, a kappa-opioid agonist with limited access to the central nervous system, has antinociceptive activity (English)

1 reference

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14 September 2022

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H. Rogers

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14 September 2022

P. J. Birch

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S. M. Harrison

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E. Palmer

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G. R. Manchee

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D. B. Judd

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A. Naylor

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D. I. Scopes

8

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A. G. Hayes

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14 September 2022

language of work or name

English

0 references

publication date

1 August 1992

1 reference

PMC publication ID

1907638

full work available at URL

15 October 2017

https://europepmc.org/articles/PMC1907638

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1327387

https://europepmc.org/articles/PMC1907638?pdf=render

14 September 2022

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1327387

British Journal of Pharmacology

14 September 2022

published in

1 reference

15 October 2017

106

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15 October 2017

4

1 reference

15 October 2017

783-789

1 reference

A kappa opioid effect: increased urination in the rat.

15 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Peripheral opioid receptors located on the rat saphenous nerve

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

16-Me cyprenorphine (RX 8008M): a potent opioid antagonist with some delta selectivity

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

In-vivo studies with the opioid antagonist, 16-methylcyprenorphine

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Antinociceptive effects of mu- and kappa-agonists in inflammation are enhanced by a peripheral opioid receptor-specific mechanism

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

ICI 204448: a kappa-opioid agonist with limited access to the CNS.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Peripheral opioid receptors mediating antinociception in inflammation. Evidence for involvement of mu, delta and kappa receptors

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Anatomy of CNS opioid receptors

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Analgesia produced by intrathecal administration of the kappa opioid agonist, U-50,488H, on formalin-evoked cutaneous pain in the rat.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Role of peripheral mu, delta and kappa opioid receptors in opioid-induced inhibition of gastrointestinal transit in rats

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Involvement of capsaicin-sensitive neurones in hyperalgesia and enhanced opioid antinociception in inflammation

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Peripheral kappa-opioid modulation of the formalin response: an electrophysiological study in the rat.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

A series of novel, highly potent and selective agonists for the kappa-opioid receptor

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

The formalin test: A quantitative study of the analgesic effects of morphine, meperidine, and brain stem stimulation in rats and cats

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

III - Prostaglandin hyperalgesia: Relevance of the peripheral effect for the analgesic action of opioid-antagonists

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Peripheral origins and central modulation of subcutaneous formalin-induced activity of rat dorsal horn neurones

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Modified formalin test: characteristic biphasic pain response

17 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

Central nervous system plasticity in the tonic pain response to subcutaneous formalin injection.

17 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1907638

The rat paw formalin test: comparison of noxious agents

17 August 2018

1 reference

12 December 2020

Opiates inhibit the discharges of fine afferent units from inflamed knee joint of the cat

1 reference

12 December 2020

Peripheral and central antinociceptive actions of ethylketocyclazocine in the formalin test

1 reference

12 December 2020

Analgesia produced by centrally administered DAGO, DPDPE and U50488H in the formalin test

1 reference

12 December 2020

Dissociation between antinociceptive and anti-inflammatory effects of acetylsalicylic acid and indomethacin in the formalin test

1 reference

12 December 2020

The formalin test in mice: dissociation between inflammatory and non-inflammatory pain

1 reference

12 December 2020

Prolonged discharge of wide-dynamic-range spinal neurons evoked by formaldehyde injected in their cutaneous receptive fields

1 reference

12 December 2020

Electrophysiological evidence for a role of bradykinin in chemical nociception in the rat

1 reference

12 December 2020

Opiate agonists inhibit neurogenic plasma extravasation in the rat

1 reference

12 December 2020

10.1111/J.1476-5381.1992.TB14413.X

Identifiers

DOI

1 reference

15 October 2017

1 reference

PMC publication ID

1907638

15 October 2017

1 reference

PMC publication ID

1907638