Novel strategies for the design of receptor-selective vasopressin analogues: Aib-substitution and retro-inverso transformation. (Q42050990)

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1 November 2019

title

Novel strategies for the design of receptor-selective vasopressin analogues: Aib-substitution and retro-inverso transformation (English)

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1 November 2019

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3

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1 November 2019

author name string

J Howl

series ordinal

1

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1 November 2019

Z Prochazka

series ordinal

2

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1 November 2019

J Slaninová

series ordinal

4

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1 November 2019

language of work or name

English

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publication date

1 October 1999

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British Journal of Pharmacology

1 November 2019

published in

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volume

128

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1 November 2019

issue

3

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1 November 2019

page(s)

647-652

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The quantitative assay of vasopressin

1 November 2019

cites work

1 reference

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Discovery of novel selective hypotensive vasopressin peptides that exhibit little or no functional interactions with known oxytocin/vasopressin receptors

5 June 2018

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Chimeric strategies for the rational design of bioactive analogs of small peptide hormones

5 June 2018

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Molecular recognition of peptide and non-peptide ligands by the extracellular domains of neurohypophysial hormone receptors

5 June 2018

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Neurohypophysial peptide systems: processing machinery, hydroosmotic regulation, adaptation and evolution

5 June 2018

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Fluorescent and biotinylated linear peptides as selective bifunctional ligands for the V1a vasopressin receptor.

5 June 2018

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Molecular cloning and functional expression of a cDNA encoding the human V1b vasopressin receptor

5 June 2018

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Molecular pharmacology of V1a vasopressin receptors.

5 June 2018

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Novel Ligand Specificity of Pituitary Vasopressin Receptors in the Rat

5 June 2018

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

5 June 2018

1 reference

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Neurohypophyseal hormone receptor systems in brain and periphery

5 June 2018

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New selective bradykinin receptor antagonists and bradykinin B2 receptor characterization

5 June 2018

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Characterization of the human liver vasopressin receptor. Profound differences between human and rat vasopressin-receptor-mediated responses suggest only a minor role for vasopressin in regulating human hepatic function

5 June 2018

1 reference

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Pharmacology and clinical perspectives of vasopressin antagonists

5 June 2018

1 reference

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A selective biotinylated probe for V1a vasopressin receptors

5 June 2018

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A radioiodinated linear vasopressin antagonist: a ligand with high affinity and specificity for V1a receptors

5 June 2018

1 reference

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Molecular cloning and expression of a rat V1a arginine vasopressin receptor

5 June 2018

1 reference

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Molecular cloning of the receptor for human antidiuretic hormone

5 June 2018

1 reference

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Potent V2/V1a vasopressin antagonists with C-terminal ethylenediamine-linked retro-amino acids

5 June 2018

1 reference

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Helix-inducing alpha-aminoisobutyric acid in opioid mimetic deltorphin C analogues

5 June 2018

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Co-evolution of ligand-receptor pairs in the vasopressin/oxytocin superfamily of bioactive peptides

17 August 2018

1 reference

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Comparison of antidiuretic and natriuretic effects of [8-lysine]vasopressin and [8-D-arginine]deaminovasopressin in conscious rats

17 August 2018

1 reference

12 December 2020

No requirement of cyclic conformation of antagonists in binding to vasopressin receptors

1 reference

12 December 2020

Novel linear antagonists of the antidiuretic (V2) and vasopressor (V1) responses to vasopressin

1 reference

12 December 2020

Pharmacological characterization of linear analogues of vasopressin generated by the systematic substitution of positions 1 and 6 by L-amino acids

1 reference

12 December 2020

Renal bradykinin and vasopressin receptors: ligand selectivity and classification

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12 December 2020

Crystal structure of a dipeptide Boc-Aib-Phe-OMe

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12 December 2020

Hormonal stimulation of phosphatidylinositol breakdown with particular reference to the hepatic effects of vasopressin

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12 December 2020

Identifiers

DOI

10.1038/SJ.BJP.0702857

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10516644%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10516644%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

PubMed publication ID

10516644

1 reference