Synthesis, modification and docking studies of 5-sulfonyl isatin derivatives as SARS-CoV 3C-like protease inhibitors (Q42250412)

24316352

19 October 2017

title

Synthesis, modification and docking studies of 5-sulfonyl isatin derivatives as SARS-CoV 3C-like protease inhibitors (English)

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19 October 2017

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Wei Liu

1

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10 June 2020

He-Min Zhu

2

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10 June 2020

Guo-Jun Niu

3

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10 June 2020

En-Zhi Shi

4

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10 June 2020

Jie Chen

5

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10 June 2020

Bo Sun

6

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10 June 2020

Wei-Qiang Chen

7

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10 June 2020

Hong-Gang Zhou

8

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10 June 2020

Cheng Yang

9

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10 June 2020

language of work or name

English

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publication date

21 November 2013

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24316352

Bioorganic & Medicinal Chemistry

19 October 2017

published in

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10 June 2020

volume

22

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10 June 2020

issue

1

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10 June 2020

page(s)

292-302

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Structure-based design and synthesis of highly potent SARS-CoV 3CL protease inhibitors

10 June 2020

cites work

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Binding interaction of quercetin-3-beta-galactoside and its synthetic derivatives with SARS-CoV 3CL(pro): structure-activity relationship studies reveal salient pharmacophore features

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Screening of electrophilic compounds yields an aziridinyl peptide as new active-site directed SARS-CoV main protease inhibitor

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SARS-CoV 3CLpro inhibitory effects of quinone-methide triterpenes from Tripterygium regelii

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Design and synthesis of peptidomimetic severe acute respiratory syndrome chymotrypsin-like protease inhibitors

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Design, synthesis, and evaluation of inhibitors for severe acute respiratory syndrome 3C-like protease based on phthalhydrazide ketones or heteroaromatic esters

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Structure-based virtual screening against SARS-3CL(pro) to identify novel non-peptidic hits

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Synthesis, docking studies, and evaluation of pyrimidines as inhibitors of SARS-CoV 3CL protease

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Synthesis of stilbene derivatives with inhibition of SARS coronavirus replication.

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Is the discovery of the novel human betacoronavirus 2c EMC/2012 (HCoV-EMC) the beginning of another SARS-like pandemic?

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Design and synthesis of new tripeptide-type SARS-CoV 3CL protease inhibitors containing an electrophilic arylketone moiety

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Synthesis of cyclopentenyl carbocyclic nucleosides as potential antiviral agents against orthopoxviruses and SARS.

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Synthesis and evaluation of isatin derivatives as effective SARS coronavirus 3CL protease inhibitors

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Synthesis and biological evaluation of nucleoside analogues having 6-chloropurine as anti-SARS-CoV agents.

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Specific Plant Terpenoids and Lignoids Possess Potent Antiviral Activities against Severe Acute Respiratory Syndrome Coronavirus

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Isatin 1,2,3-triazoles as potent inhibitors against caspase-3

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Synthesis and evaluation of pyrazolone compounds as SARS-coronavirus 3C-like protease inhibitors

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Isatin compounds as noncovalent SARS coronavirus 3C-like protease inhibitors.

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Discovery, synthesis, and structure-based optimization of a series of N-(tert-butyl)-2-(N-arylamido)-2-(pyridin-3-yl) acetamides (ML188) as potent noncovalent small molecule inhibitors of the severe acute respiratory syndrome coronavirus [...]

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Tanshinones as selective and slow-binding inhibitors for SARS-CoV cysteine proteases.

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Aryl methylene ketones and fluorinated methylene ketones as reversible inhibitors for severe acute respiratory syndrome (SARS) 3C-like proteinase

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Synthesis, crystal structure, structure-activity relationships, and antiviral activity of a potent SARS coronavirus 3CL protease inhibitor

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Identification of novel inhibitors of the SARS coronavirus main protease 3CLpro.

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12 December 2020

Design, synthesis, and evaluation of trifluoromethyl ketones as inhibitors of SARS-CoV 3CL protease

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Synthesis and activity of an octapeptide inhibitor designed for SARS coronavirus main proteinase

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12 December 2020

Coronavirus main proteinase (3CLpro) structure: basis for design of anti-SARS drugs

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12 December 2020

Design and synthesis of dipeptidyl glutaminyl fluoromethyl ketones as potent severe acute respiratory syndrome coronovirus (SARS-CoV) inhibitors

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An efficient method for the synthesis of peptide aldehyde libraries employed in the discovery of reversible SARS coronavirus main protease (SARS-CoV Mpro) inhibitors

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12 December 2020

Design, synthesis and antiviral efficacy of a series of potent chloropyridyl ester-derived SARS-CoV 3CLpro inhibitors

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Structure-based design, synthesis, and biological evaluation of peptidomimetic SARS-CoV 3CLpro inhibitors

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Potent and selective nonpeptide inhibitors of caspases 3 and 7.

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Antiviral activity of glycyrrhizic acid derivatives against SARS-coronavirus

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Synthesis and biological evaluation of quinoline salicylic acids as P-selectin antagonists

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Design and synthesis of hydroxyferroquine derivatives with antimalarial and antiviral activities.

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Design, synthesis and crystallographic analysis of nitrile-based broad-spectrum peptidomimetic inhibitors for coronavirus 3C-like proteases

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Synthesis of glutamic acid and glutamine peptides possessing a trifluoromethyl ketone group as SARS-CoV 3CL protease inhibitors

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10.1016/J.BMC.2013.11.028

Identifiers

DOI

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24316352%20AND%20SRC:MED&resulttype=core&format=json

10 June 2020

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10 June 2020

24316352

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