Agonist and inverse agonist efficacy at human recombinant serotonin 5-HT1A receptors as a function of receptor:G-protein stoichiometry (Q42441379)

31 October 2017

Agonist and inverse agonist efficacy at human recombinant serotonin 5-HT1A receptors as a function of receptor:G-protein stoichiometry (English)

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31 October 2017

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Adrian Newman-Tancredi

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31 October 2017

Conte C

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31 October 2017

Chaput C

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31 October 2017

Verrièle L

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31 October 2017

Millan MJ

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31 October 2017

1 April 1997

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31 October 2017

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36

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4-5

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451-459

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Molecular biology of 5-HT receptors

31 October 2017

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Constitutive activation of muscarinic receptors by the G-protein Gq.

7 January 2021

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Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins

7 January 2021

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Electrophysiological evidence for a large receptor reserve for inhibition of dorsal raphe neuronal firing by 5-HT1A agonists.

7 January 2021

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The genomic clone G-21 which resembles a beta-adrenergic receptor sequence encodes the 5-HT1A receptor

7 January 2021

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Electrophysiological, biochemical, neurohormonal and behavioural studies with WAY-100635, a potent, selective and silent 5-HT1A receptor antagonist

7 January 2021

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GH4ZD10 cells expressing rat 5-HT1A receptors coupled to adenylyl cyclase are a model for the postsynaptic receptors in the rat hippocampus

7 January 2021

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Interactions of purified bovine brain A1-adenosine receptors with G-proteins. Reciprocal modulation of agonist and antagonist binding.

7 January 2021

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The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro

7 January 2021

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Partial agonists, full agonists, antagonists: dilemmas of definition

7 January 2021

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Combined in situ hybridisation, northern blot analysis, and receptor binding studies in clones expressing different levels of the human 5-HT1A receptor

7 January 2021

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A serum-resistant cytofectin for cellular delivery of antisense oligodeoxynucleotides and plasmid DNA

7 January 2021

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Agonist regulation of cellular G protein levels and distribution: mechanisms and functional implications

7 January 2021

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Clozapine is a partial agonist at cloned, human serotonin 5-HT1A receptors.

7 January 2021

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S 15535 and WAY 100,635 antagonise 5-HT-stimulated [35S]GTP gamma S binding at cloned human 5-HT1A receptors

7 January 2021

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Inhibition of the constitutive activity of human 5-HT1A receptors by the inverse agonist, spiperone but not the neutral antagonist, WAY 100,635

7 January 2021

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Activity of serotonin (5-HT) receptor agonists, partial agonists and antagonists at cloned human 5-HT1A receptors that are negatively coupled to adenylate cyclase in permanently transfected HeLa cells

7 January 2021

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Cell-specific physical and functional coupling of human 5-HT1A receptors to inhibitory G protein alpha-subunits and lack of coupling to Gs alpha

7 January 2021

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Development of 5-HT1A receptor antagonists

7 January 2021

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Neurochemical profile of eltoprazine

7 January 2021

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Reverse intrinsic activity of antagonists on G protein-coupled receptors

7 January 2021

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Differentiation of NG108-15 neuroblastoma cells by serum starvation or dimethyl sulfoxide results in marked differences in angiotensin II receptor subtype expression

7 January 2021

1 reference

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Changes in G protein levels in the hippocampus and the striatum of rat brain after chronic treatment with haloperidol and sulpiride

7 January 2021

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The anti-aggressive drug eltoprazine preferentially binds to 5-HT1A and 5-HT1B receptor subtypes in rat brain: sensitivity to guanine nucleotides.

7 January 2021

1 reference

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Characterization of recombinant human serotonin 5HT1A receptors expressed in Chinese hamster ovary cells. [3H]spiperone discriminates between the G-protein-coupled and -uncoupled forms

7 January 2021

1 reference

https://api.crossref.org/works/10.1016%2FS0028-3908%2897%2900022-1

10.1016/S0028-3908(97)00022-1

7 January 2021

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31 October 2017

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