Up-regulation of a constitutively active form of the beta2-adrenoceptor by sustained treatment with inverse agonists but not antagonists (Q42528493)

1 November 2017

title

Up-regulation of a constitutively active form of the beta2-adrenoceptor by sustained treatment with inverse agonists but not antagonists (English)

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1 November 2017

MacEwan DJ

1

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1 November 2017

Milligan G

series ordinal

2

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1 November 2017

language of work or name

English

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publication date

1 December 1996

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1 November 2017

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1 November 2017

volume

399

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1 November 2017

issue

1-2

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1 November 2017

page(s)

108-112

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Reverse intrinsic activity of antagonists on G protein-coupled receptors

1 November 2017

cites work

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Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

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Agonist regulation of cellular Gs alpha-subunit levels in neuroblastoma x glioma hybrid NG108-15 cells transfected to express different levels of the human beta 2 adrenoceptor

21 January 2018

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Regulation of basal adenylate cyclase activity in neuroblastoma x glioma hybrid, NG108-15, cells transfected to express the human beta 2 adrenoceptor: evidence for empty receptor stimulation of the adenylate cyclase cascade

21 January 2018

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Foetal-calf serum stimulates a pertussis-toxin-sensitive high-affinity GTPase activity in rat glioma C6 BU1 cells

21 January 2018

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Persistent activation of the alpha subunit of Gs promotes its removal from the plasma membrane

21 January 2018

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Widespread distribution of Gq alpha/G11 alpha detected immunologically by an antipeptide antiserum directed against the predicted C-terminal decapeptide

21 January 2018

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2',5'-Dideoxyadenosine 3'-polyphosphates are potent inhibitors of adenylyl cyclases.

21 January 2018

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Chimeric alpha 2-,beta 2-adrenergic receptors: delineation of domains involved in effector coupling and ligand binding specificity

21 January 2018

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Agonist regulation of cellular G protein levels and distribution: mechanisms and functional implications

21 January 2018

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Beta 3-adrenoceptor agonist-induced down-regulation of Gs alpha and functional desensitization in a Chinese hamster ovary cell line expressing a beta 3-adrenoceptor refractory to down-regulation

21 January 2018

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Inverse agonism: pharmacological curiosity or potential therapeutic strategy?

21 January 2018

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21 January 2018

Inverse agonists exposed

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1 Assay of adenylyl cyclase catalytic activity

21 January 2018

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Constitutively active adenylyl cyclase mutant requires neither G proteins nor cytosolic regulators

21 January 2018

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Mutations of two adjacent amino acids generate inactive and constitutively active forms of the human platelet-activating factor receptor

21 January 2018

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10.1016/S0014-5793(96)01300-2

7 January 2021

Identifiers

DOI

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1 November 2017

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