Potency and selectivity of the tachykinin NK3 receptor antagonist SR 142801. (Q42551068)

2 November 2017

title

Potency and selectivity of the tachykinin NK3 receptor antagonist SR 142801. (English)

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2 November 2017

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Beaujouan JC

1

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2 November 2017

Saffroy M

series ordinal

2

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2 November 2017

Torrens Y

series ordinal

3

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2 November 2017

Glowinski J

series ordinal

4

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2 November 2017

language of work or name

English

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publication date

1 January 1997

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European Journal of Pharmacology

2 November 2017

published in

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2 November 2017

volume

319

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2 November 2017

issue

2-3

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2 November 2017

page(s)

307-316

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Neurokinin A (NK2) receptor revisited with SR 48968, a potent non-peptide antagonist

2 November 2017

cites work

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Effects of tachykinins on inositol phospholipid hydrolysis in slices of hamster urinary bladder

7 January 2021

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Molecular characterisation, expression and localisation of human neurokinin‐3 receptor

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Multiple tachykinin binding sites in hamster, rat and guinea-pig urinary bladder

7 January 2021

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The non-peptide tachykinin NK2 receptor antagonist SR 48968 interacts with human, but not rat, cloned tachykinin NK3 receptors

7 January 2021

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Phylogeny of tachykinin receptor localization in the vertebrate central nervous system: apparent absence of neurokinin-2 and neurokinin-3 binding sites in the human brain

7 January 2021

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SR 142801, the first potent non-peptide antagonist of the tachykinin NK3 receptor

7 January 2021

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The 'septide-sensitive' tachykinin receptor: still an enigma

7 January 2021

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Neurokinin3-receptors are linked to inositol phospholipid hydrolysis in the guinea-pig ileum longitudinal muscle-myenteric plexus preparation.

7 January 2021

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Pharmacological analysis of [3H]-senktide binding to NK3 tachykinin receptors in guinea-pig ileum longitudinal muscle-myenteric plexus and cerebral cortex membranes

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Receptor subtypes or species homologues: relevance to drug discovery

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Neurokinin B is a preferred agonist for a neuronal substance P receptor and its action is antagonized by enkephalin

7 January 2021

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The mammalian tachykinin receptors

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Tachykinin NK1 receptor subtypes in the rat urinary bladder.

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Two NK-3 receptor subtypes: demonstration by biological and binding assays

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Activity of SR 142801 at peripheral tachykinin receptors

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Further Demonstration that [Pro9]-Substance P Is a Potent and Selective Ligand of NK-1 Tachykinin Receptors

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The nonpeptide NK-2 antagonist SR 48968 is also a NK-3 antagonist in the guinea but not in the rat.

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7 January 2021

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Involvement of septide-sensitive tachykinin receptors in inositol phospholipid hydrolysis in the rat urinary bladder

7 January 2021

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Tissue distribution and quantitation of the mRNAs for three rat tachykinin receptors

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Specific Binding of a125I-Substance P Derivative to Rat Brain Synaptosomes

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Highly selective agonists for substance P receptor subtypes

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10.1016/S0014-2999(96)00848-5

7 January 2021

Identifiers

DOI

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2 November 2017

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