The selectivity of statine-based inhibitors against various human aspartic proteinases (Q42805724)

7 November 2017

The selectivity of statine-based inhibitors against various human aspartic proteinases (English)

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7 November 2017

Jupp RA

1

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7 November 2017

Dunn BM

2

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7 November 2017

Jacobs JW

3

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7 November 2017

Vlasuk G

4

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7 November 2017

Arcuri KE

5

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7 November 2017

Veber DF

6

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7 November 2017

Perlow DS

7

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7 November 2017

Payne LS

8

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7 November 2017

Boger J

9

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7 November 2017

de Laszlo S

10

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7 November 2017

language of work or name

English

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publication date

1 February 1990

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7 November 2017

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7 November 2017

265

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7 November 2017

3

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7 November 2017

871-878

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The determination of enzyme inhibitor constants

7 November 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

A linear equation that describes the steady-state kinetics of enzymes and subcellular particles interacting with tightly bound inhibitors

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Renin inhibitors. Syntheses of subnanomolar, competitive, transition-state analogue inhibitors containing a novel analogue of statine

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

A systematic series of synthetic chromophoric substrates for aspartic proteinases

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

On the rational design of renin inhibitors: X-ray studies of aspartic proteinases complexed with transition-state analogues

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

New inhibitors of human renin that contain novel Leu-Val replacements.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Analysis of structure-activity relationships in renin substrate analogue inhibitory peptides.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

High resolution X-ray analyses of renin inhibitor-aspartic proteinase complexes

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Synthesis and biological activity of some transition-state inhibitors of human renin

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Inhibition of porcine pepsin by two substrate analogues containing statine. The effect of histidine at the P2 subsite on the inhibition of aspartic proteinases.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Aspartic proteinases and inhibitors for their control in health and disease.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Identification of the aspartic proteinases from human erythrocyte membranes and gastric mucosa (slow-moving proteinase) as catalytically equivalent to cathepsin E

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

X-ray studies of aspartic proteinase-statine inhibitor complexes

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Effective blocking of HIV-1 proteinase activity by characteristic inhibitors of aspartic proteinases

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

In vitro inhibition of human renin by statine-containing tripeptide renin inhibitor (ES-1005)

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

CGP 38 560: orally active, low-molecular-weight renin inhibitor with high potency and specificity

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Subsite Specificity of Porcine Pepsin

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

A highly potent and long-acting oral inhibitor of human renin.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Pure human renin. Identification and characterization and of two major molecular weight forms

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

Purification and properties of cathepsin D from rat Yoshida ascites hepatoma AH-130

16 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1133712

The amino terminal amino acid sequence of human angiotensinogen

3 November 2018

1 reference

12 December 2020

Synthesis of analogues of the carboxyl protease inhibitor pepstatin. Effect of structure in subsite P3 on inhibition of pepsin

1 reference

12 December 2020

Novel renin inhibitors containing the amino acid statine

1 reference

12 December 2020

Penicillopepsin, the aspartic proteinase from Penicillium janthinellum: substrate-binding effects and intermediates in transpeptidation reactions

1 reference

12 December 2020

Design and synthesis of a potent and specific renin inhibitor with a prolonged duration of action in vivo

1 reference

12 December 2020

The pH dependence of the hydrolysis of chromogenic substrates of the type, Lys-Pro-Xaa-Yaa-Phe-(NO2)Phe-Arg-Leu, by selected aspartic proteinases: evidence for specific interactions in subsites S3 and S2

1 reference

12 December 2020

New inhibitors of human renin that contain novel Leu-Val replacements. Examination of the P1 site

1 reference

12 December 2020

New human renin inhibitors containing an unnatural amino acid, norstatine

1 reference

12 December 2020

A novel nonpeptidic, orally active renin inhibitor

1 reference

12 December 2020

The interaction of aspartic proteinases with naturally-occurring inhibitors from actinomycetes and Ascaris lumbricoides

1 reference

12 December 2020

Identifiers

DOI

10.1042/BJ2650871

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7 November 2017

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7 November 2017

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