Antiproliferative effect of a novel cholecystokinin-B/gastrin receptor antagonist, YM022. (Q42811535)

1 July 2018

title

Antiproliferative effect of a novel cholecystokinin-B/gastrin receptor antagonist, YM022. (English)

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1 July 2018

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T Murayama

1

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1 July 2018

Y Matsumori

2

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1 July 2018

N Iwata

3

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1 July 2018

M Ito

4

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1 July 2018

T Taniguchi

5

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1 July 2018

K Chihara

6

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1 July 2018

T Matsui

7

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1 July 2018

publication date

1 July 1996

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1 July 2018

number of pages

8

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Japanese Journal of Cancer Research

inferred from page(s)

published in

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1 July 2018

volume

87

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1 July 2018

issue

7

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1 July 2018

page(s)

743-750

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1 July 2018

A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists

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Tetronothiodin, a novel cholecystokinin type-B receptor antagonist produced by Streptomyces sp. NR0489. II. Isolation, characterization and biological activities

3 July 2018

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Human neuroblastoma cells express alpha and beta platelet-derived growth factor receptors coupling with neurotrophic and chemotactic signaling

3 July 2018

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Functional characterization of a human brain cholecystokinin-B receptor. A trophic effect of cholecystokinin and gastrin

3 July 2018

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Evidence for autocrine growth stimulation by a gastrin/CCK-like peptide of the gastric cancer HGT-1 cell line

3 July 2018

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Cholecystokinin Stimulates Ca2+Mobilization and Clonal Growth in Small Cell Lung Cancer through CCKAand CCKB/Gastrin Receptors

3 July 2018

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Characterization of cloned human cholecystokinin-B receptor as a gastrin receptor

3 July 2018

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Autocrine growth stimulation of human renal Wilms' tumour G401 cells by a gastrin-like peptide

3 July 2018

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Cholecystokinin-B/gastrin receptor signaling pathway involves tyrosine phosphorylations of p125FAK and p42MAP.

3 July 2018

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Antiproliferative gastrin/cholecystokinin receptor antagonists target the 78-kDa gastrin-binding protein.

3 July 2018

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Growth-promoting effects of glycine-extended progastrin

3 July 2018

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Pharmacological profile of (R)-1-[2,3-dihydro-1-(2'-methylphenacyl)-2-oxo- 5-phenyl-1H-1,4-benzodiazepin-3-yl]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin-B receptor antagonist, in vitro and in vivo

3 July 2018

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Functional characterization of two cholecystokinin-B/gastrin receptor isoforms: a preferential splice donor site in the human receptor gene

3 July 2018

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Novel gastrin receptors mediate mitogenic effects of gastrin and processing intermediates of gastrin on Swiss 3T3 fibroblasts. Absence of detectable cholecystokinin (CCK)-A and CCK-B receptors

3 July 2018

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The human brain cholecystokinin-B/gastrin receptor. Cloning and characterization

3 July 2018

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Structural analysis of the gene encoding human gastrin: the large intron contains an Alu sequence

3 July 2018

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Clinical significance of gastrin receptors in human colon cancers.

3 July 2018

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Proliferation of enterochromaffinlike cells in omeprazole-treated hypergastrinemic rats.

3 July 2018

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Independent expression of human alpha or beta platelet-derived growth factor receptor cDNAs in a naive hematopoietic cell leads to functional coupling with mitogenic and chemotactic signaling pathways

3 July 2018

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Benzodiazepine analogues L365,260 and L364,718 as gastrin and pancreatic CCK receptor antagonists

3 July 2018

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Lorglumide and loxiglumide inhibit gastrin-stimulated DNA synthesis in a rat tumoral acinar pancreatic cell line (AR42J).

3 July 2018

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Evidence for autocrine growth stimulation of cultured colon tumor cells by a gastrin/cholecystokinin-like peptide

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Pharmacological characterization of type B cholecystokinin binding sites on the human JURKAT T lymphocyte cell line.

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Partial gastric corpectomy results in hypergastrinemia and development of gastric enterochromaffinlike-cell carcinoids in the rat.

3 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Inhibitory effects of the gastrin receptor antagonist (L-365,260) on gastrointestinal tumor cells

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Interleukin-1 enhances the response of osteoblasts to platelet-derived growth factor through the alpha receptor-specific up-regulation

3 July 2018

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Therapeutic effect of the gastrin receptor antagonist, CR2093 on gastrointestinal tumour cell growth

3 July 2018

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The effect of gastrin on growth of human stomach cancer cells

3 July 2018

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Cloning and characterization of gastrin receptor from ECL carcinoid tumor of Mastomys natalensis

3 July 2018

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Expression cloning and characterization of the canine parietal cell gastrin receptor

3 July 2018

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Inhibition of gastrin-stimulated growth of gastrointestinal tumour cells by octreotide and the gastrin/cholecystokinin receptor antagonists, proglumide and lorglumide

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Gastrin stimulates Ca2+ mobilization and clonal growth in small cell lung cancer cells

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Purification, molecular cloning, and functional expression of the cholecystokinin receptor from rat pancreas

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Molecular cloning of the human brain and gastric cholecystokinin receptor: Structure, functional expression and chromosomal localization

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Differential Gene Expression of CCK(A) and CCK(B) Receptors in the Rat Brain

3 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5921164

Cholecystokinin-B/gastrin receptor: a novel molecular probe for human small cell lung cancer

16 August 2018

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12 December 2020

Effect of gastrin receptor blockade on endocrine cells in rats during achlorhydria

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12 December 2020

Antiproliferative effects of gastrin receptor antagonists and antibodies to gastrin on human colon carcinoma cell lines

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12 December 2020

Effects of gastrin and difluoromethylornithine on growth of human colon cancer

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12 December 2020

Localization of targets for anti-ulcer drugs in cells of the immune system

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12 December 2020

Enhanced hyperplasia of gastric enterochromaffinlike cells in response to omeprazole-evoked hypergastrinemia in rats with portacaval shunts. An immunocytochemical and chemical study

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12 December 2020

10.1111/J.1349-7006.1996.TB00287.X

Identifiers

DOI

1 reference

1 July 2018

PMC publication ID

5921164

1 reference

1 July 2018

PubMed publication ID

8698625

1 reference

1 July 2018