The effects of the TRPV1 receptor antagonist SB-705498 on trigeminovascular sensitisation and neurotransmission (Q43289884)

18 November 2017

The effects of the TRPV1 receptor antagonist SB-705498 on trigeminovascular sensitisation and neurotransmission (English)

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18 November 2017

6

A S Zagami

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18 November 2017

G A Lambert

1

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18 November 2017

J B Davis

2

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18 November 2017

J M Appleby

3

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18 November 2017

B A Chizh

4

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18 November 2017

K L Hoskin

5

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18 November 2017

19 August 2009

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Naunyn-Schmiedeberg's Archives of Pharmacology

18 November 2017

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18 November 2017

380

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18 November 2017

4

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18 November 2017

311-325

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https://scigraph.springernature.com/pub.10.1007/s00210-009-0437-5

18 November 2017

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https://api.crossref.org/works/10.1007%2FS00210-009-0437-5

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Randomized controlled trial of an oral CGRP receptor antagonist, MK-0974, in acute treatment of migraine

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Discovery of SB-705498: a potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development

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Evidence for a central component of post-injury pain hypersensitivity

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Nitric oxide synthase and glutamate receptor immunoreactivity in the rat spinal trigeminal neurons expressing Fos protein after formalin injection

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High affinity antagonists of the vanilloid receptor

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12 December 2020

Morphological and immunohistochemical characterization of the trigeminal ganglion neurons innervating the cornea and upper eyelid of the rat

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12 December 2020

Sensitization of meningeal sensory neurons and the origin of headaches

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12 December 2020

TRPV1 receptors in the CNS play a key role in broad-spectrum analgesia of TRPV1 antagonists

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12 December 2020

Neuropeptides and their receptors: innovative science providing novel therapeutic targets

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12 December 2020

Receptor systems mediating c-fos expression within trigeminal nucleus caudalis in animal models of migraine

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12 December 2020

Dynamic receptive field plasticity in rat spinal cord dorsal horn following C-primary afferent input

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12 December 2020

Fos expression in the trigeminocervical complex of the cat after stimulation of the superior sagittal sinus is reduced by L-NAME.

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12 December 2020

Von Frey's hairs--a review of their technology and use--a novel automated von Frey device for improved testing for hyperalgesia.

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12 December 2020

TRPV1 antagonist, SB-366791, inhibits glutamatergic synaptic transmission in rat spinal dorsal horn following peripheral inflammation

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12 December 2020

The vanilloid receptor TRPV1: 10 years from channel cloning to antagonist proof-of-concept

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12 December 2020

Characterization of SB-705498, a potent and selective vanilloid receptor-1 (VR1/TRPV1) antagonist that inhibits the capsaicin-, acid-, and heat-mediated activation of the receptor

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12 December 2020

Nitric oxide-producing islet cells modulate the release of sensory neuropeptides in the rat substantia gelatinosa

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12 December 2020

Dynamic mechanical (brush) allodynia in cluster headache

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12 December 2020

Chemical stimulation of the intracranial dura induces enhanced responses to facial stimulation in brain stem trigeminal neurons.

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The mode of action of migraine triggers: a hypothesis.

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12 December 2020

Dural vasodilation causes a sensitization of rat caudal trigeminal neurones in vivo that is blocked by a 5-HT1B/1D agonist

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12 December 2020

TRPV1 receptor mediates glutamatergic synaptic input to dorsolateral periaqueductal gray (dl-PAG) neurons.

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12 December 2020

An association between migraine and cutaneous allodynia.

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12 December 2020

Axonal transport of VR1 capsaicin receptor mRNA in primary afferents and its participation in inflammation-induced increase in capsaicin sensitivity

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12 December 2020

Cannabinoid actions on rat superficial medullary dorsal horn neurons in vitro

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12 December 2020

Activation of 5-HT(1B/1D) receptor in the periaqueductal gray inhibits nociception

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12 December 2020

Nitrergic and glutamatergic neuronal mechanisms at the trigeminovascular first-order synapse.

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12 December 2020

Terminating migraine with allodynia and ongoing central sensitization using parenteral administration of COX1/COX2 inhibitors

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Critical evaluation of the colocalization between calcitonin gene-related peptide, substance P, transient receptor potential vanilloid subfamily type 1 immunoreactivities, and isolectin B4 binding in primary afferent neurons of the rat and mouse

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12 December 2020

Distribution of mRNA for vanilloid receptor subtype 1 (VR1), and VR1-like immunoreactivity, in the central nervous system of the rat and human

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CGRP-receptor antagonists--a fresh approach to migraine therapy?

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Neuron-glia signaling in trigeminal ganglion: implications for migraine pathology

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Effect of capsaicin and resiniferatoxin on peptidergic neurons in cultured dorsal root ganglion

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Cortical blood flow changes during spreading depression in cats

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Immunohistochemical evidence for a substance P-containing trigeminovascular pathway to pial arteries in cats

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The spinal cord processing of input from the superior sagittal sinus: pathway and modulation by ergot alkaloids

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Vanilloid receptor VR1 is both presynaptic and postsynaptic in the superficial laminae of the rat dorsal horn

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12 December 2020

New migraine and pain research

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12 December 2020

Vanilloid receptor TRPV1, sensory C-fibers, and vascular autoregulation: a novel mechanism involved in myogenic constriction.

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12 December 2020

Distribution and origin of TRPV1 receptor-containing nerve fibers in the dura mater of rat.

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12 December 2020

Trigeminovascular nociceptive transmission involves N-methyl-D-aspartate and non-N-methyl-D-aspartate glutamate receptors.

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12 December 2020

Can we develop neurally acting drugs for the treatment of migraine?

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12 December 2020

Vanilloid receptor-1 (TRPV1)-dependent activation of inhibitory neurotransmission in spinal substantia gelatinosa neurons of mouse.

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12 December 2020

Is migraine a neuropathic pain syndrome?

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12 December 2020

Analgesic triptan action in an animal model of intracranial pain: a race against the development of central sensitization.

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12 December 2020

Cortico-NRM influences on trigeminal neuronal sensation

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12 December 2020

The nonpeptide calcitonin gene-related peptide receptor antagonist BIBN4096BS lowers the activity of neurons with meningeal input in the rat spinal trigeminal nucleus.

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12 December 2020

Neurogenic responses mediated by vanilloid receptor-1 (TRPV1) are blocked by the high affinity antagonist, iodo-resiniferatoxin

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12 December 2020

An immunocytochemical investigation of human trigeminal nucleus caudalis: CGRP, substance P and 5-HT1D-receptor immunoreactivities are expressed by trigeminal sensory fibres.

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12 December 2020

Autoregulation in the middle meningeal artery

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12 December 2020

Response of brainstem trigeminal neurons to electrical stimulation of the dura.

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12 December 2020

Cutaneous allodynia in transformed migraine patients

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12 December 2020

Peptidergic and serotoninergic innervation of the rat dura mater

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12 December 2020

Non-NMDA glutamate receptors modulate capsaicin induced c-fos expression within trigeminal nucleus caudalis

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12 December 2020

Comparison of responses of cutaneous nociceptive and nonnociceptive brain stem neurons in trigeminal subnucleus caudalis (medullary dorsal horn) and subnucleus oralis to natural and electrical stimulation of tooth pulp.

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12 December 2020

Immunocytochemical localization of the vanilloid receptor 1 (VR1): relationship to neuropeptides, the P2X3 purinoceptor and IB4 binding sites

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12 December 2020

The actions of anandamide on rat superficial medullary dorsal horn neurons in vitro.

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12 December 2020

Central sensitisation and cutaneous allodynia in migraine: implications for treatment

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12 December 2020

Perivascular neuropeptides (NPY, VIP, CGRP and SP) in human brain vessels after subarachnoid haemorrhage.

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12 December 2020

Capsaicin receptor immunoreactivity in the human trigeminal ganglion.

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12 December 2020

Distribution and effects of neuropeptide Y, vasoactive intestinal peptide, substance P, and calcitonin gene-related peptide in human middle meningeal arteries: Comparison with cerebral and temporal arteries

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12 December 2020

Central sensitization theory of migraine: clinical implications

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12 December 2020

NMDA-receptor activation increases cytoplasmic calcium concentration in cultured spinal cord neurones

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12 December 2020

10.1007/S00210-009-0437-5

Identifiers

DOI

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18 November 2017

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