Depressant effect on a C-fibre reflex in the rat, of RB101, a dual inhibitor of enkephalin-degrading enzymes. (Q44038445)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12079685%20AND%20SRC:MED&resulttype=core&format=json

10 November 2019

title

Depressant effect on a C-fibre reflex in the rat, of RB101, a dual inhibitor of enkephalin-degrading enzymes (English)

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10 November 2019

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4

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10 November 2019

author name string

Jean-Michel Benoist

1

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10 November 2019

Florence Keime

2

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10 November 2019

Jacqueline Montagne

3

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10 November 2019

Marie-Claude Fournié-Zaluski

5

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10 November 2019

Bernard P Roques

6

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10 November 2019

Jean-Claude Willer

7

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10 November 2019

Daniel Le Bars

8

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10 November 2019

language of work or name

English

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publication date

1 June 2002

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European Journal of Pharmacology

10 November 2019

published in

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10 November 2019

volume

445

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10 November 2019

issue

3

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10 November 2019

page(s)

201-210

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Effects of intravenous and intrathecal sufentanil on a C-fibre reflex elicited by a wide range of stimulus intensities in the rat.

10 November 2019

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Fluorescent histochemical localization of neutral endopeptidase-24.11 (enkephalinase) in the rat brainstem

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Effects of the potent analgesic enkephalin-catabolizing enzyme inhibitors RB101 and kelatorphan on respiration

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Spontaneous and evoked release of methionine-enkephalin-like material from the rat spinal cord in vivo

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Enhancement of the effects of a complete inhibitor of enkephalin-catabolizing enzymes, RB 101, by a cholecystokinin-B receptor antagonist in diabetic rats

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Prevention of degradation of endogenous enkephalins produces inhibition of nociceptive neurones in rat spinal cord

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The automated measurement of hindlimb flexor reflex of the rat as a substitute for the tail-flick assay

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A C-fiber reflex modulated by heterotopic noxious somatic stimuli in the rat

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Antinociception produced by microinjection of morphine in the rat periaqueductal gray is enhanced in the foot, but not the tail, by intrathecal injection of alpha1-adrenoceptor antagonists

7 January 2021

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Analgesic effects of kelatorphan, a new highly potent inhibitor of multiple enkephalin degrading enzymes

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"Mixed inhibitor-prodrug" as a new approach toward systemically active inhibitors of enkephalin-degrading enzymes

7 January 2021

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The distribution of nine peptides in rat spinal cord with special emphasis on the substantia gelatinosa and on the area around the central canal (laminaX)

7 January 2021

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Effects of clonidine on a C-fibre reflex in the rat

7 January 2021

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Immunohistochemical analysis of peptide pathways possibly related to pain and analgesia: enkephalin and substance P.

7 January 2021

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Enkephalin neurons that project to the A7 catecholamine cell group are located in nuclei that modulate nociception: ventromedial medulla.

7 January 2021

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Microinjection of morphine in the A7 catecholamine cell group produces opposing effects on nociception that are mediated by alpha1- and alpha2-adrenoceptors

7 January 2021

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Analgesic doses of the enkephalin degrading enzyme inhibitor RB 120 do not have discriminative stimulus properties.

7 January 2021

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7 January 2021

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Potent antinociceptive effects of kelatorphan (a highly efficient inhibitor of multiple enkephalin-degrading enzymes) systemically administered in normal and arthritic rats

7 January 2021

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Regional Metabolism of Met‐Enkephalin and Cholecystokinin on Intact Rat Brain Slices: Characterization of Specific Peptidases

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7 January 2021

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Kelatorphan potentiates the effect of [Met5]enkephalin in the substantia gelatinosa of the cat spinal cord

7 January 2021

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7 January 2021

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7 January 2021

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Unlike morphine the endogenous enkephalins protected by RB101 are unable to establish a conditioned place preference in mice

7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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7 January 2021

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inferred from DOI database lookup

7 January 2021

based on heuristic

Identifiers

DOI

10.1016/S0014-2999(02)01753-3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12079685%20AND%20SRC:MED&resulttype=core&format=json

10 November 2019

1 reference