Identification of cysteines involved in ligand binding to the human melatonin MT(2) receptor (Q44090372)

29 November 2017

title

Identification of cysteines involved in ligand binding to the human melatonin MT(2) receptor (English)

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29 November 2017

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Faika Mseeh

1

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29 November 2017

Matthew J Gerdin

series ordinal

2

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29 November 2017

Margarita I Dubocovich

series ordinal

3

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29 November 2017

language of work or name

English

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publication date

1 August 2002

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European Journal of Pharmacology

29 November 2017

published in

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29 November 2017

volume

449

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29 November 2017

issue

1-2

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29 November 2017

page(s)

29-38

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Pharmacological characterization of human recombinant melatonin mt(1) and MT(2) receptors

29 November 2017

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

7 January 2021

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The roles of valine 208 and histidine 211 in ligand binding and receptor function of the ovine Mel1a beta melatonin receptor

7 January 2021

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7 January 2021

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Role of extracellular disulfide-bonded cysteines in the ligand binding function of the beta 2-adrenergic receptor

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Selective MT2 melatonin receptor antagonists block melatonin-mediated phase advances of circadian rhythms

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The palmitoylated cysteine of the cytoplasmic tail of alpha 2A-adrenergic receptors confers subtype-specific agonist-promoted downregulation

7 January 2021

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Identification in the mu-opioid receptor of cysteine residues responsible for inactivation of ligand binding by thiol alkylating and reducing agents

7 January 2021

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Agonists induce conformational changes in transmembrane domains III and VI of the beta2 adrenoceptor

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Chimeric and point-mutated receptors reveal that a single glycine residue in transmembrane domain 6 is critical for high affinity melatonin binding.

7 January 2021

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Palmitoylation of muscarinic acetylcholine receptor m2 subtypes: reduction in their ability to activate G proteins by mutation of a putative palmitoylation site, cysteine 457, in the carboxyl-terminal tail

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7 January 2021

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7 January 2021

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A disulfide bond between conserved cysteines in the extracellular loops of the human VIP receptor is required for binding and activation

7 January 2021

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7 January 2021

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Molecular characterization of a second melatonin receptor expressed in human retina and brain: the Mel1b melatonin receptor

7 January 2021

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Melatonin receptors are for the birds: Molecular analysis of two receptor subtypes differentially expressed in chick brain

7 January 2021

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10.1016/S0014-2999(02)01903-9

7 January 2021

Identifiers

DOI

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29 November 2017

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