Synthesis and estrogen receptor affinity of a 4-hydroxytamoxifen-labeled ligand for diagnostic imaging (Q44203266)

30 November 2017

Synthesis and estrogen receptor affinity of a 4-hydroxytamoxifen-labeled ligand for diagnostic imaging (English)

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30 November 2017

Matthew R Lashley

1

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30 November 2017

Edmund J Niedzinski

2

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30 November 2017

Jane M Rogers

3

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30 November 2017

Michael S Denison

4

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30 November 2017

Michael H Nantz

5

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30 November 2017

language of work or name

English

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publication date

1 December 2002

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Bioorganic & Medicinal Chemistry

30 November 2017

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30 November 2017

10

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30 November 2017

12

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30 November 2017

4075-4082

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30 November 2017

Cancer statistics, 1999.

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Targeted anti-estrogens to treat and prevent diseases in women

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Estrogen receptor accessory proteins augment receptor-DNA interaction and DNA bending

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Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta

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The Estrogen Receptor Paradox in Breast Cancer: Association of High Receptor Concentrations with Reduced Overall Survival

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A possible divergent role for the oestrogen receptor alpha and beta subtypes in clinical breast cancer

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Differential ligand activation of estrogen receptors ERalpha and ERbeta at AP1 sites

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Determination of DNA damage in F344 rats induced by geometric isomers of tamoxifen and analogues

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Structure-activity relationships of selective estrogen receptor modulators: modifications to the 2-arylbenzothiophene core of raloxifene

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Comparative QSAR analysis of estrogen receptor ligands

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Derivatives of tamoxifen. Dependence of antiestrogenicity on the 4-substituent

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Assessing environmental chemicals for estrogenicity using a combination of in vitro and in vivo assays

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Development of high throughput screening assays using fluorescence polarization: nuclear receptor-ligand-binding and kinase/phosphatase assays

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Titration of the in vivo uptake of 16 alpha-[18F]fluoroestradiol by target tissues in the rat: competition by tamoxifen, and implications for quantitating estrogen receptors in vivo and the use of animal models in receptor-binding radiopharmaceutica

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Iodine-125-labelled tamoxifen is differentially cytoxic to cells containing oestrogen receptors

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Imaging, biodistribution and therapy potential of halogenated tamoxifen analogues

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Synthesis, biodistribution, and estrogen receptor scintigraphy of indium-111-diethylenetriaminepentaacetic acid-tamoxifen analogue

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Single isomer technetium-99m tamoxifen conjugates

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Structure, function, and regulation of androgen-binding protein/sex hormone-binding globulin

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Binding of an extracellular steroid-binding globulin to membranes and soluble receptors from human breast cancer cells (MCF-7 cells)

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Gadolinium(III) Chelates as MRI Contrast Agents: Structure, Dynamics, and Applications

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Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals

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Estrogen receptor-binding affinity of tamoxifen analogs with various side chains and their biologic profile in immature rat uterus

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Molecular basis of agonism and antagonism in the oestrogen receptor

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The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

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Efficient multigram synthesis of the bifunctional chelating agent (S)-1-p-isothiocyanatobenzyl-diethylenetriaminepentaacetic acid [correction of diethylenetetraminepentaacetic acid]

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A comparison of the inhibitory action of 5-(substituted-benzyl)-2,4-diaminopyrimidines on dihydrofolate reductase from chicken liver with that from bovine liver

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New Highly Stereoselective Synthesis of (Z)-4-Hydroxytamoxifen and (Z)-4-Hydroxytoremifene via McMurry Reaction

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Acquired tamoxifen resistance: correlation with reduced breast tumor levels of tamoxifen and isomerization of trans-4-hydroxytamoxifen.

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Structure and synthesis of dihydroxypentyluracil from bacteriophage SP-15 deoxyribonucleic acid

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Identifiers

DOI

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30 November 2017

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