Synthesis and estrogen receptor affinity of a 4-hydroxytamoxifen-labeled ligand for diagnostic imaging (Q44203266)

30 November 2017

title

Synthesis and estrogen receptor affinity of a 4-hydroxytamoxifen-labeled ligand for diagnostic imaging (English)

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30 November 2017

Matthew R Lashley

1

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30 November 2017

Edmund J Niedzinski

2

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30 November 2017

Jane M Rogers

3

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30 November 2017

Michael S Denison

4

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30 November 2017

Michael H Nantz

5

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30 November 2017

language of work or name

English

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publication date

1 December 2002

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Bioorganic & Medicinal Chemistry

30 November 2017

published in

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30 November 2017

volume

10

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30 November 2017

issue

12

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30 November 2017

page(s)

4075-4082

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30 November 2017

cites work

Cancer statistics, 1999.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Targeted anti-estrogens to treat and prevent diseases in women

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Estrogen receptor accessory proteins augment receptor-DNA interaction and DNA bending

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

The Estrogen Receptor Paradox in Breast Cancer: Association of High Receptor Concentrations with Reduced Overall Survival

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

A possible divergent role for the oestrogen receptor alpha and beta subtypes in clinical breast cancer

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Differential Ligand Activation of Estrogen Receptors ERα and ERβ at AP1 Sites

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Determination of DNA damage in F344 rats induced by geometric isomers of tamoxifen and analogues

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Structure-activity relationships of selective estrogen receptor modulators: modifications to the 2-arylbenzothiophene core of raloxifene

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Comparative QSAR analysis of estrogen receptor ligands

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Derivatives of tamoxifen. Dependence of antiestrogenicity on the 4-substituent

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Assessing environmental chemicals for estrogenicity using a combination of in vitro and in vivo assays

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Development of high throughput screening assays using fluorescence polarization: nuclear receptor-ligand-binding and kinase/phosphatase assays

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Titration of the in vivo uptake of 16 alpha-[18F]fluoroestradiol by target tissues in the rat: competition by tamoxifen, and implications for quantitating estrogen receptors in vivo and the use of animal models in receptor-binding radiopharmaceutica

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Iodine-125-labelled tamoxifen is differentially cytoxic to cells containing oestrogen receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Imaging, biodistribution and therapy potential of halogenated tamoxifen analogues

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Synthesis, biodistribution, and estrogen receptor scintigraphy of indium-111-diethylenetriaminepentaacetic acid-tamoxifen analogue

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Single isomer technetium-99m tamoxifen conjugates

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Structure, function, and regulation of androgen-binding protein/sex hormone-binding globulin

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Binding of an extracellular steroid-binding globulin to membranes and soluble receptors from human breast cancer cells (MCF-7 cells)

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Gadolinium(III) Chelates as MRI Contrast Agents: Structure, Dynamics, and Applications

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Estrogen receptor-binding affinity of tamoxifen analogs with various side chains and their biologic profile in immature rat uterus

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Molecular basis of agonism and antagonism in the oestrogen receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Efficient multigram synthesis of the bifunctional chelating agent (S)-1-p-isothiocyanatobenzyl-diethylenetriaminepentaacetic acid [correction of diethylenetetraminepentaacetic acid]

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

A comparison of the inhibitory action of 5-(substituted-benzyl)-2,4-diaminopyrimidines on dihydrofolate reductase from chicken liver with that from bovine liver

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

New Highly Stereoselective Synthesis of (Z)-4-Hydroxytamoxifen and (Z)-4-Hydroxytoremifene via McMurry Reaction

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Acquired tamoxifen resistance: correlation with reduced breast tumor levels of tamoxifen and isomerization of trans-4-hydroxytamoxifen.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Structure and synthesis of dihydroxypentyluracil from bacteriophage SP-15 deoxyribonucleic acid

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

Conjugation of antibodies with bifunctional chelating agents: isothiocyanate and bromoacetamide reagents, methods of analysis, and subsequent addition of metal ions

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2802%2900329-2

7 January 2021

10.1016/S0968-0896(02)00329-2

Identifiers

DOI

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30 November 2017

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