A homology-based model of the human 5-HT2A receptor derived from an in silico activated G-protein coupled receptor (Q44268642)

1 December 2017

A homology-based model of the human 5-HT2A receptor derived from an in silico activated G-protein coupled receptor (English)

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G protein-coupled receptor

1 December 2017

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author name string

James J Chambers

series ordinal

1

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PubMed ID

12510883

1 December 2017

David E Nichols

series ordinal

2

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PubMed ID

12510883

1 December 2017

language of work or name

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1 July 2002

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Journal of Computer - Aided Molecular Design

1 December 2017

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1 December 2017

16

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1 December 2017

7

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1 December 2017

511-520

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https://scigraph.springernature.com/pub.10.1023/a:1021275430021

1 December 2017

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cites work

Rhodopsin: a prototypical G protein-coupled receptor

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12 December 2020

Formation of the meta II photointermediate is accompanied by conformational changes in the cytoplasmic surface of rhodopsin

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12 December 2020

Fourier transform infrared difference spectra of intermediates in rhodopsin bleaching

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12 December 2020

Photoelectron spectra of psychotropic drugs. 6. Relationships between physical properties and pharmacological actions of amphetamine analogs

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Contribution of a helix 5 locus to selectivity of hallucinogenic and nonhallucinogenic ligands for the human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors: direct and indirect effects on ligand affinity mediated by the same locus

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12 December 2020

Requirement of rigid-body motion of transmembrane helices for light activation of rhodopsin

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Resolution and absolute configuration of trans-2-(2,5-dimethoxy-4-methylphenyl)cyclopropylamine, a potent hallucinogen analog

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Further studies on oxygenated tryptamines with LSD-like activity incorporating a chiral pyrrolidine moiety into the side chain

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Conformational changes in rhodopsin probed by surface plasmon resonance spectroscopy

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12 December 2020

Enantiospecific synthesis and pharmacological evaluation of a series of super-potent, conformationally restricted 5-HT(2A/2C) receptor agonists

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12 December 2020

Species differences in the pharmacology of the 5-hydroxytryptamine2 receptor: structurally specific differentiation by ergolines and tryptamines

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12 December 2020

Study of global motions in proteins by weighted masses molecular dynamics: adenylate kinase as a test case.

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12 December 2020

Comparative protein modelling by satisfaction of spatial restraints

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12 December 2020

Structure and function of serotonin 5-HT2 receptors

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Activation of rhodopsin: new insights from structural and biochemical studies

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Using CLUSTAL for multiple sequence alignments

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12 December 2020

Photoactivated conformational changes in rhodopsin: a time-resolved spin label study

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12 December 2020

Receptors and G proteins as primary components of transmembrane signal transduction. Part 1. G-protein-coupled receptors: structure and function.

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Crystal structure of rhodopsin: A G protein-coupled receptor

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12 December 2020

Fourier transform infrared spectroscopy indicates a major conformational rearrangement in the activation of rhodopsin.

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Areas, volumes, packing and protein structure

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12 December 2020

The role of conserved aspartate and serine residues in ligand binding and in function of the 5-HT1A receptor: a site-directed mutation study

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1-(2,5-Dimethoxy-4-(trifluoromethyl)phenyl)-2-aminopropane: a potent serotonin 5-HT2A/2C agonist

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12 December 2020

Species variations in transmembrane region V of the 5-hydroxytryptamine type 2A receptor alter the structure-activity relationship of certain ergolines and tryptamines

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12 December 2020

N(1)-substituted ergolines and tryptamines show species differences for the agonist-labeled 5-HT2 receptor.

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12 December 2020

A geometric approach to macromolecule-ligand interactions

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12 December 2020

Mapping the binding site pocket of the serotonin 5-Hydroxytryptamine2A receptor. Ser3.36(159) provides a second interaction site for the protonated amine of serotonin but not of lysergic acid diethylamide or bufotenin

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Constitutive activation of opsin: influence of charge at position 134 and size at position 296.

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12 December 2020

Specific tryptophan UV-absorbance changes are probes of the transition of rhodopsin to its active state

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12 December 2020

Identifiers

DOI

10.1023/A:1021275430021

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journals/jcamd/ChambersN02

1 December 2017

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DBLP Dataset 2021-01-02

Dimensions Publication ID

28 January 2021

0 references

1 reference

PubMed ID

12510883