Bias Factor and Therapeutic Window Correlate to Predict Safer Opioid Analgesics (Q44351142)

2 December 2017

title

Bias Factor and Therapeutic Window Correlate to Predict Safer Opioid Analgesics (English)

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2 December 2017

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Cullen L Schmid

1

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2 December 2017

Nicole M Kennedy

2

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2 December 2017

Nicolette C Ross

3

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2 December 2017

Kimberly M Lovell

4

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2 December 2017

Zhizhou Yue

5

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2 December 2017

Jenny Morgenweck

6

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2 December 2017

Michael D Cameron

7

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2 December 2017

Thomas D Bannister

8

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2 December 2017

Laura M Bohn

9

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2 December 2017

language of work or name

English

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publication date

1 November 2017

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2 December 2017

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2 December 2017

volume

171

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2 December 2017

issue

5

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2 December 2017

page(s)

1165-1175.e13

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Addressing the Fentanyl Threat to Public Health

2 December 2017

cites work

1 reference

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Biased agonism of the μ-opioid receptor by TRV130 increases analgesia and reduces on-target adverse effects versus morphine: A randomized, double-blind, placebo-controlled, crossover study in healthy volunteers

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27 August 2018

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A G protein-biased ligand at the μ-opioid receptor is potently analgesic with reduced gastrointestinal and respiratory dysfunction compared with morphine

27 August 2018

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14-Alkoxy- and 14-acyloxypyridomorphinans: μ agonist/δ antagonist opioid analgesics with diminished tolerance and dependence side effects

27 August 2018

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27 August 2018

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Agonist-directed interactions with specific beta-arrestins determine mu-opioid receptor trafficking, ubiquitination, and dephosphorylation.

27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

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27 August 2018

1 reference

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27 August 2018

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Bezitramide (R 4845), a new potent and orally long-acting analgesic compound

27 August 2018

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27 August 2018

1 reference

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inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.CELL.2017.10.035

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2 December 2017

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