Prolylisoxazoles: potent inhibitors of prolyloligopeptidase with antitrypanosomal activity (Q44651596)

5 December 2017

title

Prolylisoxazoles: potent inhibitors of prolyloligopeptidase with antitrypanosomal activity (English)

1 reference

5 December 2017

2

1 reference

5 December 2017

4

1 reference

5 December 2017

7

1 reference

5 December 2017

5

Philippe Grellier

1 reference

5 December 2017

Gunther Bal

1

1 reference

5 December 2017

Dimitri Antonov

series ordinal

3

1 reference

5 December 2017

Simon L Croft

series ordinal

6

1 reference

5 December 2017

Achiel Haemers

series ordinal

8

1 reference

5 December 2017

language of work or name

English

0 references

publication date

1 September 2003

1 reference

Bioorganic & Medicinal Chemistry Letters

5 December 2017

published in

1 reference

5 December 2017

volume

13

1 reference

5 December 2017

issue

17

1 reference

5 December 2017

page(s)

2875-2878

1 reference

Proline specific peptidases

5 December 2017

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

A Trypanosoma cruzi-secreted 80 kDa proteinase with specificity for human collagen types I and IV.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Identification of inhibitors of an 80 kDa protease from Trypanosoma cruzi through the screening of a combinatorial peptide library

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Automated parallel synthesis of a tetrahydroisoquinolin-based library: potential prolyl endopeptidase inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Synthesis and activity of pyrrolidinyl- and thiazolidinyl-dipeptide derivatives as inhibitors of the Tc80 prolyl oligopeptidase from Trypanosoma cruzi

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Comparison of the inhibition of human and Trypanosoma cruzi prolyl endopeptidases

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Trypanosoma cruzi prolyl oligopeptidase Tc80 is involved in nonphagocytic mammalian cell invasion by trypomastigotes.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Synthesis, structure-activity relationships, and pharmacokinetic profiles of nonpeptidic alpha-keto heterocycles as novel inhibitors of human chymase.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Peptidyl alpha-ketoheterocyclic inhibitors of human neutrophil elastase. 2. Effect of varying the heterocyclic ring on in vitro potency

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Synthesis and structure-activity relationships of peptidyl alpha-keto heterocycles as novel inhibitors of prolyl endopeptidase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Prolyl Oligopeptidase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

The Reactions of Primary Nitroparaffins with Isocyanates1

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

The Henry reaction: recent examples

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

An Efficient Synthesis of Optically Active α-(t-Butoxycarbonylamino)-aldehydes from α-Amino Acids

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Oxidation of Alcohols by Activated Dimethyl Sulfoxide and Related Reactions: An Update

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Frontier molecular orbitals of 1,3 dipoles and dipolarophiles

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Development and evaluation of peptide-based prolyl oligopeptidase inhibitors--introduction of N-benzyloxycarbonyl-prolyl-3-fluoropyrrolidine as a lead in inhibitor design.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

An in-vitro system for determining the activity of compounds against the intracellular amastigote form of Leishmania donovani

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

Efficient technique for screening drugs for activity against Trypanosoma cruzi using parasites expressing beta-galactosidase

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

The Alamar Blue assay to determine drug sensitivity of African trypanosomes (T.b. rhodesiense and T.b. gambiense) in vitro

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2803%2900579-1

7 January 2021

10.1016/S0960-894X(03)00579-1

Identifiers

DOI

1 reference

5 December 2017

1 reference