In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. (Q45351488)

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scientific article published on 22 May 2008

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English	In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity.	scientific article published on 22 May 2008

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scholarly article

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7 January 2020

In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity (English)

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7 January 2020

8

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7 January 2020

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Simona Bertoni

1

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7 January 2020

Vigilio Ballabeni

2

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7 January 2020

Lisa Flammini

3

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7 January 2020

Francesca Saccani

4

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7 January 2020

Giuseppe Domenichini

5

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7 January 2020

Giovanni Morini

6

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7 January 2020

Mara Comini

7

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7 January 2020

Elisabetta Barocelli

9

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7 January 2020

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22 May 2008

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7 January 2020

Naunyn-Schmiedeberg's Archives of Pharmacology

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7 January 2020

378

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7 January 2020

3

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7 January 2020

335-343

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7 January 2020

Medicinal chemistry and biological properties of non-imidazole histamine H3 antagonists

1 reference

https://api.crossref.org/works/10.1007%2FS00210-008-0299-2

21 January 2018

Anticholinesterase activity--studies on chemical models. 5. Symmetrical bisquarternary cyclic amines with a rigid interquarternary chain

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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Acute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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Discovery of histamine H3 receptor antagonistic property of simple imidazole-free derivatives: Preliminary pharmacological investigation

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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Rapid colorimetric assay for cell growth and survival. Modifications to the tetrazolium dye procedure giving improved sensitivity and reliability

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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The first potent and selective non-imidazole human histamine H4 receptor antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

based on heuristic

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Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

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Multiple enzyme inhibitions by histamine H3 receptor antagonists as potential procognitive agents.

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

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Dibasic non-imidazole histamine H3 receptor antagonists with a rigid biphenyl scaffold

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

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The histamine H3 receptor: from gene cloning to H3 receptor drugs

1 reference

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12 December 2020

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Pharmacological profile of new thioperamide derivatives at histamine peripheral H1-, H2-, H3-receptors in guinea-pig

1 reference

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12 December 2020

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

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Histamine H3 receptor antagonists: preclinical promise for treating obesity and cognitive disorders

1 reference

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12 December 2020

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Inhibition and induction of cytochrome P450 and the clinical implications

1 reference

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12 December 2020

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A new class of diamine-based human histamine H3 receptor antagonists: 4-(aminoalkoxy)benzylamines

1 reference

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12 December 2020

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GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models

1 reference

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12 December 2020

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Interactions of new and conventional H3-antagonists with non-histaminergic receptors involved in neurogenic and myogenic contractile responses of guinea-pig ileum

1 reference

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12 December 2020

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Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists: in vitro properties, drug-likeness, and behavioral activity

1 reference

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12 December 2020

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In vivo occupancy of histamine H3 receptors by thioperamide and (R)-alpha-methylhistamine measured using histamine turnover and an ex vivo labeling technique

1 reference

https://pubmed.ncbi.nlm.nih.gov/18496672

12 December 2020

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Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow

1 reference

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12 December 2020

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Cumulative dose-response curves. II. Technique for the making of dose-response curves in isolated organs and the evaluation of drug parameters

1 reference

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In vitro pharmacology at human histamine H3 receptors and brain access of non-imidazole alkylpiperidine derivatives

1 reference

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Modulation of neurotransmitter release via histamine H3 heteroreceptors

1 reference

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12 December 2020

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Effects of histamine H3 receptor agonists and antagonists on cognitive performance and scopolamine-induced amnesia.

1 reference

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A new and rapid colorimetric determination of acetylcholinesterase activity

1 reference

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Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas

1 reference

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12 December 2020

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Identifiers

10.1007/S00210-008-0299-2

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18496672%20AND%20SRC:MED&resulttype=core&format=json

7 January 2020

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18496672%20AND%20SRC:MED&resulttype=core&format=json

7 January 2020

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