Dose-dependent sigma-1 receptor occupancy by donepezil in rat brain can be assessed with (11)C-SA4503 and microPET. (Q45663984)

15 December 2017

title

Dose-dependent sigma-1 receptor occupancy by donepezil in rat brain can be assessed with (11)C-SA4503 and microPET. (English)

1 reference

15 December 2017

Nisha K Ramakrishnan

1

1 reference

15 December 2017

Anniek K D Visser

2

1 reference

15 December 2017

Marianne Schepers

3

1 reference

15 December 2017

Gert Luurtsema

4

1 reference

15 December 2017

Csaba J Nyakas

5

1 reference

15 December 2017

Philip H Elsinga

6

1 reference

15 December 2017

Kiichi Ishiwata

7

1 reference

15 December 2017

Rudi A J O Dierckx

8

1 reference

15 December 2017

Aren van Waarde

9

1 reference

15 December 2017

language of work or name

1 reference

18 March 2014

1 reference

15 December 2017

1 reference

15 December 2017

volume

231

1 reference

15 December 2017

issue

20

1 reference

15 December 2017

page(s)

3997-4006

1 reference

https://scigraph.springernature.com/pub.10.1007/s00213-014-3533-2

15 December 2017

exact match

0 references

cites work

Safety, tolerability and pharmacokinetics of single and multiple doses of a novel sigma-1 receptor antagonist in three randomized phase I studies

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Degree of inhibition of cortical acetylcholinesterase activity and cognitive effects by donepezil treatment in Alzheimer's disease.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Measuring drug occupancy in the absence of a reference region: the Lassen plot re-visited

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Dopamine D2 occupancy as a biomarker for antipsychotics: quantifying the relationship with efficacy and extrapyramidal symptoms

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Evidence that the potential antipsychotic agent rimcazole (BW 234U) is a specific, competitive antagonist of sigma sites in brain

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Brain levels and acetylcholinesterase inhibition with galantamine and donepezil in rats, mice, and rabbits

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Pharmacokinetic and pharmacodynamic properties of cholinesterase inhibitors donepezil, tacrine, and galantamine in aged and young Lister hooded rats.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Donepezil (E2020): a new acetylcholinesterase inhibitor. Review of its pharmacology, pharmacokinetics, and utility in the treatment of Alzheimer's disease

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Procognitive 5-HT6 antagonists in the rat forced swimming test: potential therapeutic utility in mood disorders associated with Alzheimer's disease.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

High occupancy of sigma1 receptors in the human brain after single oral administration of donepezil: a positron emission tomography study using [11C]SA4503.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Regional response of cerebral blood volume to graded hypoxic hypoxia in rat brain

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Regional effects of donepezil and rivastigmine on cortical acetylcholinesterase activity in Alzheimer's disease

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

TAK-147, an acetylcholinesterase inhibitor, increases choline acetyltransferase activity in cultured rat septal cholinergic neurons

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Synthesis and evaluation of 11C- and 18F-labeled 1-[2-(4-alkoxy-3-methoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazines as sigma receptor ligands for positron emission tomography studies

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Phencyclidine-induced cognitive deficits in mice are ameliorated by subsequent subchronic administration of donepezil: role of sigma-1 receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Donepezil primarily attenuates scopolamine-induced deficits in psychomotor function, with moderate effects on simple conditioning and attention, and small effects on working memory and spatial mapping.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Sigma 1 receptor subtype is involved in the relief of behavioral despair in the mouse forced swimming test

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Interaction with sigma(1) protein, but not N-methyl-D-aspartate receptor, is involved in the pharmacological activity of donepezil

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Interactions of selective serotonin reuptake inhibitors with subtypes of sigma receptors in rat brain

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Concurrent administration of atypical antipsychotics and donepezil: drug interaction study in rats.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Small-animal PET with a σ-ligand, 11C-SA4503, detects spontaneous pituitary tumors in aged rats.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Mapping of human cerebral sigma1 receptors using positron emission tomography and [11C]SA4503.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

A template for spatial normalisation of MR images of the rat brain

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Effect of donepezil on brain acetylcholinesterase activity in patients with AD measured by PET.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Sigma opiates and certain antipsychotic drugs mutually inhibit (+)-[3H] SKF 10,047 and [3H]haloperidol binding in guinea pig brain membranes

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

The cholinergic system, sigma-1 receptors and cognition

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Sigma receptors in oncology: therapeutic and diagnostic applications of sigma ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Pharmacological interaction with the sigma1 (σ1)-receptor in the acute behavioral effects of antidepressants.

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Anti-dementia drugs and hippocampal-dependent memory in rodents

21 January 2018

1 reference

https://api.crossref.org/works/10.1007%2FS00213-014-3533-2

Involvement of the sigma1 receptor in the antidepressant-like effects of fluvoxamine in the forced swimming test in comparison with the effects elicited by paroxetine

21 January 2018

1 reference

12 December 2020

Benzodiazepine Receptor Quantification in vivo in Humans Using [11C]Flumazenil and PET: Application of the Steady-State Principle

1 reference

12 December 2020

Inhibitory effects of donepezil hydrochloride (E2020) on cholinesterase activity in brain and peripheral tissues of young and aged rats

1 reference

12 December 2020

Limited donepezil inhibition of acetylcholinesterase measured with positron emission tomography in living Alzheimer cerebral cortex.

1 reference

12 December 2020

10.1007/S00213-014-3533-2

Identifiers

DOI

1 reference

Dimensions Publication ID

15 December 2017

1053303393

0 references

1 reference