A fluorometric screening assay for drug efflux transporter activity in the blood-brain barrier (Q46382844)

21 December 2017

title

A fluorometric screening assay for drug efflux transporter activity in the blood-brain barrier (English)

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21 December 2017

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Corbin J Bachmeier

1

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21 December 2017

Donald W Miller

series ordinal

2

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21 December 2017

publication date

1 January 2005

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21 December 2017

published in

Pharmaceutical Research

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21 December 2017

volume

22

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21 December 2017

issue

1

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21 December 2017

page(s)

113-121

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21 December 2017

Multidrug resistance protein-mediated transport of chlorambucil and melphalan conjugated to glutathione

cites work

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Crossref

https://api.crossref.org/works/10.1007%2FS11095-004-9016-0

Transport properties of the multidrug resistance-associated protein (MRP) in human tumour cells

21 January 2018

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12 December 2020

Hyperthermia, cyclosporine A and melphalan cytotoxicity and transport in multidrug resistant cells

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12 December 2020

Drug efflux transport properties of 2',7'-bis(2-carboxyethyl)-5(6)-carboxyfluorescein acetoxymethyl ester (BCECF-AM) and its fluorescent free acid, BCECF.

1 reference

12 December 2020

Expression of various multidrug resistance-associated protein (MRP) homologues in brain microvessel endothelial cells

1 reference

12 December 2020

P-glycoprotein in the blood-brain barrier of mice influences the brain penetration and pharmacological activity of many drugs

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12 December 2020

In vitro and in vivo reversal of multidrug resistance by GF120918, an acridonecarboxamide derivative.

1 reference

12 December 2020

Distribution of multi-drug resistance-associated P-glycoprotein in normal and neoplastic human tissues. Analysis with 3 monoclonal antibodies recognizing different epitopes of the P-glycoprotein molecule

1 reference

12 December 2020

Characterization of the regional intestinal kinetics of drug efflux in rat and human intestine and in Caco-2 cells

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12 December 2020

Effects of MDR1 and MDR3 P-glycoproteins, MRP1, and BCRP/MXR/ABCP on the transport of (99m)Tc-tetrofosmin

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12 December 2020

Pluronic P85 increases permeability of a broad spectrum of drugs in polarized BBMEC and Caco-2 cell monolayers.

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12 December 2020

Characterization of the human multidrug resistance protein isoform MRP3 localized to the basolateral hepatocyte membrane

1 reference

12 December 2020

Coordinated action of glutathione S-transferases (GSTs) and multidrug resistance protein 1 (MRP1) in antineoplastic drug detoxification. Mechanism of GST A1-1- and MRP1-associated resistance to chlorambucil in MCF7 breast carcinoma cells

1 reference

12 December 2020

In vitro P-glycoprotein affinity for atypical and conventional antipsychotics

1 reference

12 December 2020

Transport of amphipathic anions by human multidrug resistance protein 3

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12 December 2020

Secretion of organic anions by hepatocytes: involvement of homologues of the multidrug resistance protein.

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12 December 2020

Effect of GF120918, a potent P-glycoprotein inhibitor, on morphine pharmacokinetics and pharmacodynamics in the rat

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12 December 2020

Use of rhodamine 123 to examine the functional activity of P-glycoprotein in primary cultured brain microvessel endothelial cell monolayers

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12 December 2020

Tissue and cell distribution of the multidrug resistance-associated protein (MRP) in mouse intestine and kidney

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12 December 2020

Role of multidrug resistance protein 1 (MRP1) and glutathione S-transferase A1-1 in alkylating agent resistance. Kinetics of glutathione conjugate formation and efflux govern differential cellular sensitivity to chlorambucil versus melphalan toxicit

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12 December 2020

Tissue distribution of P-glycoprotein encoded by a multidrug-resistant gene as revealed by a monoclonal antibody, MRK 16

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12 December 2020

Subcellular localization and distribution of the breast cancer resistance protein transporter in normal human tissues.

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12 December 2020

Reversal of resistance by GF120918 in cell lines expressing the ABC half-transporter, MXR.

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12 December 2020

Selective inhibition of MDR1 P-glycoprotein-mediated transport by the acridone carboxamide derivative GG918.

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12 December 2020

Plasma membrane localization of multidrug resistance-associated protein homologs in brain capillary endothelial cells

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12 December 2020

The effect of hyperthermia and verapamil on melphalan cytotoxicity and transport in multidrug-resistant Chinese hamster ovary cells

1 reference

12 December 2020

Rational use of in vitro P-glycoprotein assays in drug discovery

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12 December 2020

Cellular localization of the multidrug-resistance gene product P-glycoprotein in normal human tissues

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12 December 2020

Serum Concentrations and Side Effects in Psychiatric Patients During Risperidone Therapy

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12 December 2020

Localisation of breast cancer resistance protein in microvessel endothelium of human brain

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12 December 2020

A multidrug resistance transporter from human MCF-7 breast cancer cells

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12 December 2020

Multidrug-resistance gene (P-glycoprotein) is expressed by endothelial cells at blood-brain barrier sites

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12 December 2020

Characterisation of the brain multidrug resistance protein (BMDP/ABCG2/BCRP) expressed at the blood–brain barrier

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12 December 2020

A family of drug transporters: the multidrug resistance-associated proteins.

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12 December 2020

Analysis of expression of cMOAT (MRP2), MRP3, MRP4, and MRP5, homologues of the multidrug resistance-associated protein gene (MRP1), in human cancer cell lines

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12 December 2020

Interaction of morphine, fentanyl, sufentanil, alfentanil, and loperamide with the efflux drug transporter P-glycoprotein

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12 December 2020

Expression of MDR1 (multidrug resistance) gene and its protein in normal human kidney

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12 December 2020

Transepithelial transport of nicotine and vinblastine in isolated malpighian tubules of the tobacco hornworm (Manduca sexta) suggests a P-glycoprotein-like mechanism

1 reference

12 December 2020

Expression of the multidrug resistance gene product (P-glycoprotein) in human normal and tumor tissues.

1 reference

12 December 2020

MDR1 gene expression: its effect on drug resistance to doxorubicin in human hepatocellular carcinoma cell lines.

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12 December 2020

Cellular efflux pump and interaction between cisplatin and paclitaxel in ovarian cancer cells

1 reference

12 December 2020

Characterization of multidrug resistance by fluorescent dyes.

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12 December 2020

Taxol: mechanisms of action and resistance.

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12 December 2020

A new multidrug resistance protein at the blood-brain barrier

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12 December 2020

Mammalian drug efflux transporters of the ATP binding cassette (ABC) family: an overview.

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12 December 2020

Valproic acid uptake by bovine brain microvessel endothelial cells: role of active efflux transport.

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12 December 2020

P-glycoprotein expression by cancer cells affects cell cytotoxicity and cell-cycle perturbations induced by six chemotherapeutic drugs

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12 December 2020

Involvement of multidrug resistance associated protein 1 (Mrp1) in the efflux transport of 17beta estradiol-D-17beta-glucuronide (E217betaG) across the blood-brain barrier

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12 December 2020

P-glycoprotein-mediated efflux transport of anticancer drugs at the blood-brain barrier.

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12 December 2020

Role of transporters in the tissue-selective distribution and elimination of drugs: transporters in the liver, small intestine, brain and kidney

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12 December 2020

Expression of multidrug resistance-associated protein (MRP) in brain microvessel endothelial cells.

1 reference

12 December 2020

Effects of a potent and specific P-glycoprotein inhibitor on the blood-brain barrier distribution and antinociceptive effect of morphine in the rat.

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12 December 2020

Antifolate resistance mediated by the multidrug resistance proteins MRP1 and MRP2.

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12 December 2020

Characterization of efflux transport of organic anions in a mouse brain capillary endothelial cell line

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12 December 2020

A putative nicotine pump at the metabolic blood-brain barrier of the tobacco hornworm

1 reference

12 December 2020

The multidrug-resistant phenotype associated with overexpression of the new ABC half-transporter, MXR (ABCG2)

1 reference

12 December 2020

Effect of P-glycoprotein modulation on the clinical pharmacokinetics and adverse effects of morphine

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12 December 2020

10.1007/S11095-004-9016-0

Identifiers

DOI

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21 December 2017

release_5dlalah46fdthaqub72x24n3ti

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/5dlalah46fdthaqub72x24n3ti

24 November 2022

mapped directly with Wikidata item

PubMed ID

15771237

1 reference

21 December 2017