Development of a BRET2 screening assay using beta-arrestin 2 mutants (Q47360713)

14 January 2018

title

Development of a BRET2 screening assay using beta-arrestin 2 mutants (English)

1 reference

14 January 2018

author name string

Milka Vrecl

1

1 reference

14 January 2018

Rasmus Jorgensen

2

1 reference

14 January 2018

Azra Pogacnik

3

1 reference

14 January 2018

Anders Heding

4

1 reference

14 January 2018

publication date

1 June 2004

1 reference

14 January 2018

Journal of Biomolecular Screening

published in

1 reference

14 January 2018

volume

9

1 reference

14 January 2018

issue

4

1 reference

14 January 2018

page(s)

322-333

1 reference

14 January 2018

Target validation of G-protein coupled receptors

cites work

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Designing screens: how to make your hits a hit.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Endocytosis of G protein-coupled receptors: roles of G protein-coupled receptor kinases and beta-arrestin proteins

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Arresting developments in heptahelical receptor signaling and regulation

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Differential affinities of visual arrestin, beta arrestin1, and beta arrestin2 for G protein-coupled receptors delineate two major classes of receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Molecular determinants underlying the formation of stable intracellular G protein-coupled receptor-beta-arrestin complexes after receptor endocytosis*

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Arrestin/clathrin interaction. Localization of the arrestin binding locus to the clathrin terminal domain

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

The beta2-adrenergic receptor/betaarrestin complex recruits the clathrin adaptor AP-2 during endocytosis

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

The interaction of beta-arrestin with the AP-2 adaptor is required for the clustering of beta 2-adrenergic receptor into clathrin-coated pits

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

beta-Arrestin/AP-2 interaction in G protein-coupled receptor internalization: identification of a beta-arrestin binging site in beta 2-adaptin

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Recent advances in technology for measuring and manipulating cell signals

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

A bioluminescence resonance energy transfer (BRET) system: application to interacting circadian clock proteins

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Dimerization: an emerging concept for G protein-coupled receptor ontogeny and function

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

The BRET2/arrestin assay in stable recombinant cells: a platform to screen for compounds that interact with G protein-coupled receptors (GPCRS).

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Applications of novel resonance energy transfer techniques to study dynamic hormone receptor interactions in living cells.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

The use of resonance energy transfer in high-throughput screening: BRET versus FRET.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Homo- and hetero-oligomeric interactions between G-protein-coupled receptors in living cells monitored by two variants of bioluminescence resonance energy transfer (BRET): hetero-oligomers between receptor subtypes form more efficiently than between

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Novel method for the study of receptor Ca2+ signalling exemplified by the NK1 receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Modeling of sequestration and down regulation in cells containing beta2-adrenergic receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

The cellular distribution of fluorescently labeled arrestins provides a robust, sensitive, and universal assay for screening G protein-coupled receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Conservation of the phosphate-sensitive elements in the arrestin family of proteins

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Differential roles of arrestin-2 interaction with clathrin and adaptor protein 2 in G protein-coupled receptor trafficking

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Scaffolding functions of arrestin-2 revealed by crystal structure and mutagenesis

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Crystal structure of beta-arrestin at 1.9 A: possible mechanism of receptor binding and membrane Translocation

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Heterologous regulation of trafficking and signaling of G protein-coupled receptors: beta-arrestin-dependent interactions between neurokinin receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Identification of a novel human eicosanoid receptor coupled to G(i/o)

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Novel detection strategies for drug discovery

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Association of beta-arrestin with G protein-coupled receptors during clathrin-mediated endocytosis dictates the profile of receptor resensitization

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Targeted construction of phosphorylation-independent beta-arrestin mutants with constitutive activity in cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Desensitization of the neurokinin-1 receptor (NK1-R) in neurons: effects of substance P on the distribution of NK1-R, Galphaq/11, G-protein receptor kinase-2/3, and beta-arrestin-1/2

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Substance P-induced trafficking of beta-arrestins. The role of beta-arrestins in endocytosis of the neurokinin-1 receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

The nature of the arrestin x receptor complex determines the ultimate fate of the internalized receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Role of beta-arrestin in mediating agonist-promoted G protein-coupled receptor internalization

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

Constitutive and agonist-dependent homo-oligomerization of the thyrotropin-releasing hormone receptor. Detection in living cells using bioluminescence resonance energy transfer

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057104263212

21 January 2018

Identifiers

DOI

10.1177/1087057104263212

1 reference

14 January 2018

1 reference

14 January 2018