Species selectivity of nonpeptide antagonists of the gonadotropin-releasing hormone receptor is determined by residues in extracellular loops II and III and the amino terminus (Q47448039)

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scientific article published on 21 May 2004

Language	Label	Description	Also known as
English	Species selectivity of nonpeptide antagonists of the gonadotropin-releasing hormone receptor is determined by residues in extracellular loops II and III and the amino terminus	scientific article published on 21 May 2004

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scholarly article

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

Species selectivity of nonpeptide antagonists of the gonadotropin-releasing hormone receptor is determined by residues in extracellular loops II and III and the amino terminus (English)

1 reference

Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

author name string

Greg J Reinhart

1

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

Qiu Xie

2

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

Xin-Jun Liu

3

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

Yun-Fei Zhu

4

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PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

Jun Fan

5

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Europe PubMed Central

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16 January 2018

http://europepmc.org/abstract/MED/15155770

Chen Chen

6

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

R Scott Struthers

7

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

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publication date

21 May 2004

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

number of pages

8

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Journal of Biological Chemistry

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16 January 2018

http://europepmc.org/abstract/MED/15155770

279

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16 January 2018

http://europepmc.org/abstract/MED/15155770

33

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16 January 2018

http://europepmc.org/abstract/MED/15155770

34115-34122

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Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequence

1 reference

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Primary structure of the ovine hypothalamic luteinizing hormone-releasing factor (LRF) (LH-hypothalamus-LRF-gas chromatography-mass spectrometry-decapeptide-Edman degradation).

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21 January 2018

Uncovering molecular mechanisms involved in activation of G protein-coupled receptors

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Molecular mechanisms of ligand interaction with the gonadotropin-releasing hormone receptor

1 reference

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Progress towards the development of non-peptide orally-active gonadotropin-releasing hormone (GnRH) antagonists: therapeutic implications.

1 reference

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Synthesis and initial structure-activity relationships of a novel series of imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists

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Design, synthesis and structure-activity relationships of novel imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists

1 reference

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Initial structure-activity relationship studies of a novel series of pyrrolo[1,2-a]pyrimid-7-ones as GnRH receptor antagonists

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Synthesis and structure-activity relationships of 1-arylmethyl-3-(2-aminopropyl)-5-aryl-6-methyluracils as potent GnRH receptor antagonists

1 reference

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21 January 2018

Species differences in the sensitivity to a GnRH antagonist

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M404474200

21 January 2018

Gonadotropin-releasing hormone analog design. Structure-function studies toward the development of agonists and antagonists: rationale and perspective

1 reference

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21 January 2018

Design and Structure−Activity Relationships of 2-Alkyl-3-aminomethyl-6-(3-methoxyphenyl)-7-methyl-8-(2-fluorobenzyl)imidazolo[1,2-a]pyrimid-5-ones as Potent GnRH Receptor Antagonists

1 reference

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21 January 2018

Crystal structure of rhodopsin: A G protein-coupled receptor

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

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21 January 2018

The biologically crucial C terminus of cholecystokinin and the non-peptide agonist SR-146,131 share a common binding site in the human CCK1 receptor. Evidence for a crucial role of Met-121 in the activation process

1 reference

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21 January 2018

Tyrosine 220 in the 5th transmembrane domain of the neuromedin B receptor is critical for the high selectivity of the peptoid antagonist PD168368.

1 reference

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21 January 2018

Structural requirements for the activation of the human growth hormone secretagogue receptor by peptide and nonpeptide secretagogues

1 reference

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21 January 2018

Mutagenesis and modeling of the neurotensin receptor NTR1. Identification of residues that are critical for binding SR 48692, a nonpeptide neurotensin antagonist

1 reference

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21 January 2018

Irreversible activation of the gonadotropin-releasing hormone receptor by photoaffinity cross-linking: localization of attachment site to Cys residue in N-terminal segment

1 reference

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21 January 2018

A new photoreactive antagonist cross-links to the N-terminal domain of the gonadotropin-releasing hormone receptor

1 reference

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21 January 2018

Two Mutations in Extracellular Loop 2 of the Human GnRH Receptor Convert an Antagonist to an Agonist

1 reference

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21 January 2018

Identifiers

10.1074/JBC.M404474200

1 reference

Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

16 January 2018

http://europepmc.org/abstract/MED/15155770

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