Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors. (Q47738911)

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scientific article published in December 2017

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English	Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors.	scientific article published in December 2017

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26 March 2020

Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors (English)

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26 March 2020

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26 March 2020

Ramin Ekhteiari Salmas

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26 March 2020

Claudiu T Supuran

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Claudiu T Supuran

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26 March 2020

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Belma Zengin Kurt

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26 March 2020

Fatih Sonmez

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26 March 2020

Busecan Aksoydan

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26 March 2020

Mustafa Kucukislamoglu

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26 March 2020

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1 December 2017

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26 March 2020

Journal of Enzyme Inhibition and Medicinal Chemistry

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26 March 2020

32

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26 March 2020

1

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26 March 2020

1042-1052

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26 March 2020

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Creative Commons Attribution 4.0 International

1 January 2017

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April 2022 Public Data File from Crossref

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April 2022 Public Data File from Crossref

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Design of a Carbonic Anhydrase IX Active-Site Mimic To Screen Inhibitors for Possible Anticancer Properties † ‡

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Carbonic Anhydrase: Structure, Catalytic Versatility, and Inhibition

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12 December 2020

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Design and synthesis of coumarin-3-acylamino derivatives to scavenge radicals and to protect DNA

1 reference

https://pubmed.ncbi.nlm.nih.gov/28776440

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Carbonic anhydrase inhibitors. Arylsulfonylureido- and arylureido-substituted aromatic and heterocyclic sulfonamides: towards selective inhibitors of carbonic anhydrase isozyme I

1 reference

https://pubmed.ncbi.nlm.nih.gov/28776440

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII

1 reference

https://pubmed.ncbi.nlm.nih.gov/28776440

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The expression of carbonic anhydrase II in hematological malignancies

1 reference

https://pubmed.ncbi.nlm.nih.gov/28776440

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Discovery of potent carbonic anhydrase and acetylcholine esterase inhibitors: novel sulfamoylcarbamates and sulfamides derived from acetophenones

1 reference

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based on heuristic

inferred from PubMed ID database lookup

Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XII

1 reference

https://pubmed.ncbi.nlm.nih.gov/28776440

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based on heuristic

inferred from PubMed ID database lookup

Interaction of carbonic anhydrase isozymes I, II, and IX with some pyridine and phenol hydrazinecarbothioamide derivatives

1 reference

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based on heuristic

inferred from PubMed ID database lookup

Dendrimers incorporating benzenesulfonamide moieties strongly inhibit carbonic anhydrase isoforms I-XIV

1 reference

https://pubmed.ncbi.nlm.nih.gov/28776440

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

New aminobenzenesulfonamide-thiourea conjugates: synthesis and carbonic anhydrase inhibition and docking studies

1 reference

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based on heuristic

inferred from PubMed ID database lookup

Acetylcholinesterase and carbonic anhydrase inhibitory properties of novel urea and sulfamide derivatives incorporating dopaminergic 2-aminotetralin scaffolds

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1080/14756366.2017.1354857

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28776440%20AND%20SRC:MED&resulttype=core&format=json

26 March 2020

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28776440%20AND%20SRC:MED&resulttype=core&format=json

26 March 2020

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28776440%20AND%20SRC:MED&resulttype=core&format=json

26 March 2020

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