Radioreceptor binding reveals the potencies of N,N-disubstituted 2-aminotetralins as D2 dopamine agonists (Q48190385)

9 February 2018

title

Radioreceptor binding reveals the potencies of N,N-disubstituted 2-aminotetralins as D2 dopamine agonists (English)

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9 February 2018

author name string

P M Beart

1

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9 February 2018

C J Cook

2

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9 February 2018

M Cincotta

3

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9 February 2018

D J de Vries

4

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9 February 2018

P Tepper

5

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9 February 2018

D Dijkstra

6

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9 February 2018

A S Horn

7

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9 February 2018

publication date

1 November 1987

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9 February 2018

Naunyn-Schmiedeberg's Archives of Pharmacology

published in

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9 February 2018

volume

336

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9 February 2018

issue

5

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9 February 2018

page(s)

487-493

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9 February 2018

Synthesis and radioreceptor binding activity of N-0437, a new, extremely potent and selective D2 dopamine receptor agonist

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N-0434, a very potent and specific new D-2 dopamine receptor agonist

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High-and Low-Affinity States of Striatal D2Receptors Are Not Affected by 6-Hydroxydopamine or Chronic Haloperidol Treatment

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The guanine nucleotide activating site of the regulatory component of adenylate cyclase. Identification by ligand binding

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N,N-disubstituted 2-aminotetralins are potent D-2 dopamine receptor agonists

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Role of assay conditions in determining agonist potency at D2 dopamine receptors in striatal homogenates

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8-Hydroxy-2-(di-n-propylamino)tetralin, a new centrally acting 5-hydroxytryptamine receptor agonist

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The ternary complex model. Its properties and application to ligand interactions with the D2-dopamine receptor of the anterior pituitary gland

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Guanine nucleotides reveal differential actions of ergot derivatives at D-2 receptors labelled by [3H]spiperone in striatal homogenates

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Kinetic and pharmacological profiles of the in vitro binding of the potent dopamine agonist [3H]N,N-dipropyl-5,6-dihydroxy-2-aminotetralin to rat striatal membranes

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Effect of non-catecholic 2-aminotetralin derivatives on dopamine metabolism in the rat striatum

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Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes

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The role of D-1 and D-2 receptors

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Agonist high- and low-affinity states of the D2-dopamine receptor in calf brain. Partial conversion by guanine nucleotide

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In vivo dopamine autoreceptor selectivity appears to be critically dependent upon the aromatic hydroxyl position in a series of N,N-disubstituted 2-aminotetralins

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Dopamine receptor model and its application in the design of a new class of rigid pyrrolo[2,3-g]isoquinoline antipsychotics

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Biochemical Properties of Hormone-Sensitive Adenylate Cyclase

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A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor

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Dopamine inhibition of anterior pituitary adenylate cyclase is mediated through the high-affinity state of the D2 receptor

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Dopaminergic inhibition of adenylate cyclase correlates with high affinity agonist binding to anterior pituitary D2 dopamine receptors

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Identifiers

DOI

10.1007/BF00169304

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9 February 2018

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9 February 2018