High throughput artificial membrane permeability assay for blood-brain barrier (Q48349894)

10 February 2018

title

High throughput artificial membrane permeability assay for blood-brain barrier (English)

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10 February 2018

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Li Di

1

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10 February 2018

Edward H Kerns

2

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10 February 2018

Kristi Fan

3

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10 February 2018

Oliver J McConnell

4

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10 February 2018

Guy T Carter

5

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10 February 2018

publication date

1 March 2003

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10 February 2018

European Journal of Medicinal Chemistry

published in

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10 February 2018

volume

38

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10 February 2018

issue

3

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10 February 2018

page(s)

223-232

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10 February 2018

Computational methods for the prediction of 'drug-likeness'

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Multivariate pharmaceutical profiling for drug discovery

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The functional role of P-glycoprotein in the blood-brain barrier

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7 January 2021

Transporter-mediated permeation of drugs across the blood-brain barrier

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7 January 2021

Relationship of octanol/water partition coefficient and molecular weight to rat brain capillary permeability

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7 January 2021

Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists

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7 January 2021

Potential of immobilized artificial membranes for predicting drug penetration across the blood-brain barrier

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7 January 2021

Rapid calculation of polar molecular surface area and its application to the prediction of transport phenomena. 2. Prediction of blood-brain barrier penetration

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7 January 2021

Correlation and prediction of a large blood-brain distribution data set--an LFER study

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7 January 2021

Molecular factors influencing drug transfer across the blood-brain barrier

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7 January 2021

Blood-brain barrier permeation: molecular parameters governing passive diffusion

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7 January 2021

A method to determine the ability of drugs to diffuse through the blood-brain barrier

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7 January 2021

Hydrogen bonding. 33. Factors that influence the distribution of solutes between blood and brain.

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7 January 2021

Computation of brain-blood partitioning of organic solutes via free energy calculations

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7 January 2021

Theoretical calculation and prediction of brain-blood partitioning of organic solutes using MolSurf parametrization and PLS statistics

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7 January 2021

Physicochemical high throughput screening: parallel artificial membrane permeation assay in the description of passive absorption processes

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7 January 2021

High-throughput permeability pH profile and high-throughput alkane/water log P with artificial membranes

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7 January 2021

A comparative study of artificial membrane permeability assay for high throughput profiling of drug absorption potential

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7 January 2021

Predicting blood-brain barrier permeation from three-dimensional molecular structure.

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7 January 2021

Transport into retina measured by short vascular perfusion in the rat.

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7 January 2021

Blood-brain barrier transport of caffeine: dose-related restriction of adenine transport

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7 January 2021

Transport of protein-bound hormones into tissues in vivo

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7 January 2021

The effects of atenolol (tenormin) and methyldopa on simple tests of central nervous function

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7 January 2021

Quinolone therapy for infections of the central nervous system

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7 January 2021

Blood-to-brain transfer of various oxicams: effects of plasma binding on their brain delivery

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7 January 2021

Lipid and fatty acyl composition of rat brain capillary endothelia isolated by a new technique

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7 January 2021

Cortisol is transported by the multidrug resistance gene product P-glycoprotein

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7 January 2021

P-glycoprotein in the blood-brain barrier of mice influences the brain penetration and pharmacological activity of many drugs

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7 January 2021

Cardiotoxic effect with convulsions in terfenadine overdose

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7 January 2021

Interplay between CYP3A-mediated metabolism and polarized efflux of terfenadine and its metabolites in intestinal epithelial Caco-2 (TC7) cell monolayers

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7 January 2021

Quantum Calculation of Molecular Energies and Energy Gradients in Solution by a Conductor Solvent Model

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7 January 2021

10.1016/S0223-5234(03)00012-6

Identifiers

DOI

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10 February 2018

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10 February 2018