NCQ 298, a new selective iodinated salicylamide ligand for the labelling of dopamine D2 receptors (Q48827053)

15 February 2018

title

NCQ 298, a new selective iodinated salicylamide ligand for the labelling of dopamine D2 receptors (English)

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25 October 2022

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25 October 2022

dopaminergic

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25 October 2022

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25 October 2022

3

C Halldin

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15 February 2018

author name string

H. Hall

1

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25 October 2022

T. Högberg

2

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25 October 2022

C. Köhler

4

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25 October 2022

P. Ström

5

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25 October 2022

S. B. Ross

6

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S. A. Larsson

7

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L. Farde

8

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25 October 2022

language of work or name

English

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National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=1672460

25 October 2022

publication date

1 January 1991

1 reference

15 February 2018

full work available at URL

http://link.springer.com/content/pdf/10.1007/BF02244067.pdf

file format

Portable Document Format

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http://link.springer.com/article/10.1007/BF02244067/fulltext.html

25 October 2022

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http://link.springer.com/content/pdf/10.1007/BF02244067

25 October 2022

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25 October 2022

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15 February 2018

volume

103

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15 February 2018

issue

1

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15 February 2018

page(s)

6-18

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15 February 2018

Central D2-dopamine receptor occupancy in schizophrenic patients treated with antipsychotic drugs

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Quantitative analysis of drug-receptor interactions: I. Determination of kinetic and equilibrium properties

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Dopamine D2 receptors in the cerebral cortex: distribution and pharmacological characterization with [3H]raclopride

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Autoradiographic visualization of dopamine D-2 receptors in the monkey brain using the selective benzamide drug [3H]raclopride

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Sodium-dependent isomerization of dopamine D-2 receptors characterized using [125I]epidepride, a high-affinity substituted benzamide ligand.

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Generalized scatter correction method in SPECT using point scatter distribution functions.

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The absolute density of neurotransmitter receptors in the brain. Example for dopamine receptors

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Dopamine D-2 receptor imaging radiopharmaceuticals: synthesis, radiolabeling, and in vitro binding of (R)-(+)- and (S)-(-)-3-iodo-2-hydroxy-6-methoxy-N- [(1-ethyl-2-pyrrolidinyl)methyl]benzamide

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Effects of chronic neuroleptic treatment on agonist affinity states of the dopamine-D2 receptor in the rat brain

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Preparation and biodistribution of [125I]IBZM: a potential CNS D-2 dopamine receptor imaging agent

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Contamination of serotonin-2 binding sites by an alpha-1 adrenergic component in assays with (3H) spiperone

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Gamma camera emission tomography. Development and properties of a multi-sectional emission computed tomography system

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Imaging dopamine receptors in the human brain by positron tomography

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3HRo 22-1319 (piquindone) binds to the D2 dopaminergic receptor subtype in a sodium-dependent manner

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Potential neuroleptic agents. 3. Chemistry and antidopaminergic properties of substituted 6-methoxysalicylamides

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Syntheses of [123I]-, [125I]- and unlabelled (S)-3-iodo-5,6-dimethoxy-N-[(1-ethyl-2-pyrrolidinyl)methyl]salicylamide (NCQ 298), selective ligands for the study of dopamine D-2 receptors.

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Stereoselective binding of 11C-raclopride in living human brain--a search for extrastriatal central D2-dopamine receptors by PET.

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Characteristics of [3H]sultopride binding to rat brain.

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Uptake of 77Br-spiperone in the striata of schizophrenic patients and controls

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12 December 2020

Nuclear medicine: SPECT comparisons to PET.

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Kinetic analysis of central [11C]raclopride binding to D2-dopamine receptors studied by PET--a comparison to the equilibrium analysis

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A special cut-off gamma camera for high-resolution SPECT of the head.

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Quantitative analysis of D2 dopamine receptor binding in the living human brain by PET.

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Antipsychotic drug doses and neuroleptic/dopamine receptors

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Serotonergic component of neuroleptic receptors

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Spiperone: a ligand of choice for neuroleptic receptors. 1. Kinetics and characteristics of in vitro binding

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Cation regulation differentiates specific binding of [3 H]sulpiride and [3 H]spiperone to rat striatal preparations

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[125I]iodopride: a specific high affinity radioligand for labelling striatal dopamine D-2 receptors.

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Effects of temperature on the in vitro binding of 3H-raclopride to rat striatal dopamine-D2 receptors

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Specific in vitro and in vivo binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain

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Kinetic properties of the accumulation of 3H-raclopride in the mouse brain in vivo

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Endogenous dopamine lowers the dopamine D2 receptor density as measured by [3H]raclopride: implications for positron emission tomography of the human brain

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New selective dopamine D-2 antagonists as antipsychotic agents. Pharmacological, chemical, structural and theoretical considerations

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In vivo labelling of rat brain dopamine D-2 receptors. Stereoselective blockade by the D-2 antagonist raclopride and its enantiomer of 3H-spiperone, 3H-N,N-propylnorapomorphine and 3H-raclopride binding in the rat brain

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12 December 2020

Potential neuroleptic agents. 4. Chemistry, behavioral pharmacology, and inhibition of [3H]spiperone binding of 3,5-disubstituted N-[(1-ethyl-2-pyrrolidinyl)methyl]-6-methoxysalicylamides

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12 December 2020

The selective dopamine D2 receptor antagonist raclopride discriminates between dopamine-mediated motor functions.

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12 December 2020

Carbon-11 labelling of eticlopride in two different positions--a selective high-affinity ligand for the study of dopamine D-2 receptors using PET

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12 December 2020

1,3-Di(2-[5-3H]tolyl)guanidine: a selective ligand that labels sigma-type receptors for psychotomimetic opiates and antipsychotic drugs

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12 December 2020

[125]I-spectramide: a novel benzamide displaying potent and selective effects at the D2 dopamine receptor.

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12 December 2020

Comparisons between the in vitro binding of two substituted benzamides and two butyrophenones to dopamine-D2 receptors in the rat striatum

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12 December 2020

Potential antipsychotic agents. 7. Synthesis and antidopaminergic properties of the atypical highly potent (S)-5-bromo-2,3-dimethoxy-N-[(1-ethyl-2-pyrrolidinyl)methyl]benzamide and related compounds. A comparative study.

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Some in vitro receptor binding properties of [3H]eticlopride, a novel substituted benzamide, selective for dopamine-D2 receptors in the rat brain

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Comparison of the in vitro receptor binding properties of N-[3H]methylspiperone and [3H]raclopride to rat and human brain membranes.

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12 December 2020

Substituted benzamides as ligands for visualization of dopamine receptor binding in the human brain by positron emission tomography

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Potential antipsychotic agents 5. Synthesis and antidopaminergic properties of substituted 5,6-dimethoxysalicylamides and related compounds

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Brain dopamine receptors

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Effects of remoxipride and some related new substituted salicylamides on rat brain receptors.

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12 December 2020

Evaluation of a semiautomatic filtration technique for receptor binding studies

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Acta pharmaceutica Suecica

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Identifiers

DOI

10.1007/BF02244067

1 reference

15 February 2018

1 reference

15 February 2018