Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV (Q57480761)

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scholarly article by Noriyasu Kato et al published December 2011 in Bioorganic & Medicinal Chemistry
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English
Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV
scholarly article by Noriyasu Kato et al published December 2011 in Bioorganic & Medicinal Chemistry

    Statements

    Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV (English)
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    Noriyasu Kato
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    Mitsuru Oka
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    Takayo Murase
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    Masahiro Yoshida
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    Masao Sakairi
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    Satoko Yamashita
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    Yoshika Yasuda
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    Aya Yoshikawa
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    Yuuji Hayashi
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    Mitsuhiro Makino
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    Motohiro Takeda
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    Yakufu Mirensha
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    Takuji Kakigami
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    December 2011
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    19
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    7221-7227
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    23
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