Rational design of dynorphin A analogues with δ-receptor selectivity and antagonism for δ- and κ-receptors (Q57951338)

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10 November 2019

title

Rational design of dynorphin A analogues with delta-receptor selectivity and antagonism for delta- and kappa-receptors (English)

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10 November 2019

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1

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10 November 2019

Anna Capasso

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10 November 2019

Severo Salvadori

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10 November 2019

author name string

M Marastoni

3

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10 November 2019

S D Bryant

4

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10 November 2019

P S Cooper

5

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10 November 2019

L H Lazarus

6

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10 November 2019

P A Temussi

7

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10 November 2019

language of work or name

English

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publication date

1 January 1998

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Bioorganic & Medicinal Chemistry

10 November 2019

published in

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10 November 2019

volume

6

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10 November 2019

issue

1

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10 November 2019

page(s)

57-62

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Identification of two related pentapeptides from the brain with potent opiate agonist activity

10 November 2019

cites work

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Morphine-like ligand for opiate receptors in human CSF

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Isolation of an endogenous compound from the brain with pharmacological properties similar to morphine

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

A potent and selective endogenous agonist for the mu-opiate receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Managing post-herpetic neuralgia with opioids and local anesthetics

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Naloxone reduces the neurochemical and behavioral effects of amphetamine but not those of cocaine.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Kappa-opioids produce significantly greater analgesia in women than in men.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Synthesis and opioid activity of 2-substituted dynorphin A-(1-13) amide analogues

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Synthesis and opioid activity of dynorphin A-(1-13)NH2 analogues containing cis- and trans-4-aminocyclohexanecarboxylic acid

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Synthesis and Opioid Activity of Conformationally Constrained Dynorphin A Analogs. 1. Conformational Constraint in the "Message" Sequence

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

The opioid peptides of the amphibian skin

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Function of negative charge in the "address domain" of deltorphins

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Stereospecificity of amino acid side chains in deltorphin defines binding to opioid receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Conformationally restricted deltorphin analogues

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Phe3-substituted analogues of deltorphin C. Spatial conformation and topography of the aromatic ring in peptide recognition by delta opioid receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Morphiceptin (NH 4 -Tyr-Pro-Phe-Pro-COHN 2 ): a Potent and Specific Agonist for Morphine (μ) Receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Conversion of enkephalin and dermorphin into delta-selective opioid antagonists by single-residue substitution.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Selective opioid dipeptides

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Evolution of the Dmt-Tic pharmacophore: N-terminal methylated derivatives with extraordinary delta opioid antagonist activity

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Systemic analgesic activity and delta-opioid selectivity in [2,6-dimethyl-Tyr1,D-Pen2,D-Pen5]enkephalin

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Analogs of the delta opioid receptor selective cyclic peptide [2-D-penicillamine,5-D-penicillamine]-enkephalin: 2',6'-dimethyltyrosine and Gly3-Phe4 amide bond isostere substitutions

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Preparation and opioid activity of analogues of the analgesic dipeptide 2,6-dimethyl-L-tyrosyl-N-(3-phenylpropyl)-D-alaninamide

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Opioid receptor selectivity alteration by single residue replacement: synthesis and activity profile of [Dmt1]deltorphin B.

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Dermorphin analogues carrying an increased positive net charge in their "message" domain display extremely high mu opioid receptor selectivity

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Differentiation between rat brain and mouse vas deferens delta opioid receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Sequence of kappa-opioid receptor cDNA in the R1.1 thymoma cell line

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Structure and expression of a rat kappa opioid receptor gene

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Difluorotoluene, a Nonpolar Isostere for Thymine, Codes Specifically and Efficiently for Adenine in DNA Replication

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Design and solution structure of a partially rigid opioid antagonist lacking the basic center--models of antagonism

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

Synthesis and biological activities of dynorphin A analogues with opioid antagonist properties

1 reference

https://api.crossref.org/works/10.1016%2FS0968-0896%2897%2910008-6

7 January 2021

10.1016/S0968-0896(97)10008-6

Identifiers

DOI

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10 November 2019

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