Piperidinylpyrroles: Design, synthesis and binding properties of novel and selective dopamine D4 receptor ligands (Q64030247)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10560741%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

title

Piperidinylpyrroles: design, synthesis and binding properties of novel and selective dopamine D4 receptor ligands (English)

1 reference

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1 November 2019

main subject

drug discovery

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pharmaceutical science

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author

Peter Gmeiner

series ordinal

3

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10560741%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

author name string

C Haubmann

series ordinal

1

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10560741%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

H Hübner

series ordinal

2

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10560741%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

language of work or name

English

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publication date

1 November 1999

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10560741%20AND%20SRC:MED&resulttype=core&format=json

1 November 2019

number of pages

4

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Bioorganic & Medicinal Chemistry Letters

inferred from page(s)

published in

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1 November 2019

volume

9

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1 November 2019

issue

21

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1 November 2019

page(s)

3143-3146

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Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine

1 November 2019

cites work

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Dopamine D4 receptors elevated in schizophrenia

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3-((4-(4-Chlorophenyl)piperazin-1-yl)-methyl)-1H-pyrrolo-2,3-b-pyridine: an antagonist with high affinity and selectivity for the human dopamine D4 receptor

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7 January 2021

Azaindole derivatives with high affinity for the dopamine D4 receptor: Synthesis, ligand binding studies and comparison of molecular electrostatic potential maps

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1-Phenyl-3-(aminomethyl)pyrroles as potential antipsychotic agents. Synthesis and dopamine receptor binding

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7 January 2021

2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors

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7 January 2021

SAR of novel biarylmethylamine dopamine D4 receptor ligands

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7 January 2021

5-(4-Chlorophenyl)-4-methyl-3-(1-(2-phenylethyl)piperidin-4-yl)isoxazole: a potent, selective antagonist at human cloned dopamine D4 receptors

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7 January 2021

4-Heterocyclylpiperidines as selective high-affinity ligands at the human dopamine D4 receptor

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7 January 2021

4-N-linked-heterocyclic piperidine derivatives with high affinity and selectivity for human dopamine D4 receptors

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7 January 2021

1-(3-Cyanobenzylpiperidin-4-yl)-5-methyl-4-phenyl-1, 3-dihydroimidazol-2-one: a selective high-affinity antagonist for the human dopamine D(4) receptor with excellent selectivity over ion channels

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7 January 2021

2,2-dicyanovinyl as a nonaromatic aryl bioisostere: synthesis, binding experiments and SAR studies of highly selective dopamine D4 receptor ligands

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7 January 2021

Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor

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7 January 2021

Modulation of Intracellular Cyclic AMP Levels by Different Human Dopamine D4 Receptor Variants

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7 January 2021

Enantio- and diastereocontrolled dopamine D1, D2, D3 and D4 receptor binding of N-(3-pyrrolidinylmethyl)benzamides synthesized from aspartic acid

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7 January 2021

10.1016/S0960-894X(99)00540-5

Identifiers

DOI

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1 November 2019

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